SCHEMBL26465843

SCHEMBL26465843

O=C(CN1CC2CC(C1)N2CC1(F)CCC(F)(F)CC1)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
KDM4E B2RXH2 1/20 0.46
CACNA1H O95180 10/20 0.44
LMNA P02545 1/20 0.40
THRB P10828 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PSMB5 P28074 1/20 0.40
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
EPHX1 P07099 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26465828 0.90 ALDH1A1 (0.48) ALDH1A1KDM4ECACNA1HLMNATHRB
SCHEMBL26465831 0.78 ALDH1A1 (0.50) ALDH1A1KDM4ECACNA1HPSMB5
SCHEMBL26466619 0.74 ALDH1A1 (0.43) ALDH1A1KDM4ECACNA1HLMNATHRB
SCHEMBL26465830 0.74 CACNA1H (0.73) ALDH1A1KDM4ECACNA1HPSMB5KMT2A
SCHEMBL26465978 0.73 KDM4E (0.45) ALDH1A1KDM4ECACNA1HPSMB5MEN1
SCHEMBL26465836 0.72 CACNA1H (0.56) ALDH1A1KDM4ECACNA1HPSMB5EPHX1
SCHEMBL26465834 0.70 MEN1 (0.48) ALDH1A1KDM4ECACNA1HPSMB5MEN1
SCHEMBL26463801 0.68 CACNA1H (0.71) ALDH1A1KDM4ECACNA1HKMT2A
SCHEMBL26466782 0.68 KDM4E (0.42) ALDH1A1KDM4ECACNA1HPSMB5MAPT
SCHEMBL4217027 0.68 ALDH1A1 (0.60) ALDH1A1KDM4ECACNA1HPSMB5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192669-A1 T-TYPE CALCIUM CHANNEL MODULATORS COMPRISING A PIPERAZINE OR 1,4-DIAZEPANE CORE AND METHODS OF USE THEREOF PRAXIS PRECISION MEDICINES, INC. (US) 2023-10-05 WO disclosed