SCHEMBL26484643

SCHEMBL26484643

CC(=O)c1ccn(Cc2ccc3ccccc3c2)c(=O)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
CTRB1 P17538 1/20 0.41
MAPK14 Q16539 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
DAO P14920 1/20 0.40
HPGD P15428 1/20 0.40
CYP19A1 P11511 1/20 0.40
MMP13 P45452 1/20 0.39
MCHR1 Q99705 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21650581 0.88 KMT2A (0.47) CTRB1MAPK14MEN1KMT2AMCHR1
SCHEMBL31066573 0.86 CTRB1 (0.55) CTRB1MAPK14DAO
SCHEMBL31066580 0.86 POLB (0.46) ALDH1A1MEN1KMT2AMCHR1
SCHEMBL21634096 0.86 POLB (0.46) ALDH1A1MEN1KMT2AMCHR1
SCHEMBL12640061 0.84 MAPK14 (0.52) MAPK14
SCHEMBL21634140 0.84 NPC1 (0.48) ALDH1A1MAPTCTRB1NPC1MMP13
SCHEMBL31066644 0.84 NPC1 (0.48) ALDH1A1MAPTCTRB1NPC1MMP13
SCHEMBL20503971 0.77 FLT1 (0.48) ALDH1A1MAPK14KMT2ADAOCYP19A1
SCHEMBL17457967 0.76 KMT2A (0.51) KMT2ADAOCYP19A1
SCHEMBL12734354 0.73 ACACB (0.42) MAPTMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3827004-B1 4-(1,3,4-OXADIAZOLE-2-YL)PYRIDINE-2(1H)-ONE DERIVATIVES AS HISTONE DEACETYLASE 6 (HDAC6) INHIBITORS FOR THE TREATMENT OF E.G. INFECTIONS CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2023-10-11 EP disclosed