SCHEMBL21650581

SCHEMBL21650581

O=C(O)c1ccn(Cc2ccc3ccccc3c2)c(=O)c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
MEN1 O00255 1/20 0.47
TBXAS1 P24557 1/20 0.47
MCHR1 Q99705 1/20 0.45
PTGER4 P35408 2/20 0.45
PTGER2 P43116 2/20 0.45
MAPK14 Q16539 1/20 0.45
NR1H4 Q96RI1 1/20 0.44
MRGPRX4 Q96LA9 2/20 0.43
CYP1A2 P05177 1/20 0.42
CTRB1 P17538 1/20 0.42
FAAH O00519 1/20 0.41
PTPN1 P18031 1/20 0.41
ACP1 P24666 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26484643 0.88 ALDH1A1 (0.42) KMT2AMEN1MCHR1MAPK14CTRB1
SCHEMBL31066573 0.88 CTRB1 (0.55) MAPK14CTRB1FAAH
SCHEMBL31066644 0.85 NPC1 (0.48) MCHR1NR1H4CTRB1
SCHEMBL21634140 0.85 NPC1 (0.48) MCHR1NR1H4CTRB1
SCHEMBL1255936 0.85 MAPK14 (0.55) KMT2AMEN1MAPK14
SCHEMBL21634096 0.84 POLB (0.46) KMT2AMEN1MCHR1FAAH
SCHEMBL31066580 0.84 POLB (0.46) KMT2AMEN1MCHR1FAAH
SCHEMBL14576364 0.80 MAPK8 (0.48) KMT2AMEN1MAPK14MRGPRX4
SCHEMBL20503971 0.78 FLT1 (0.48) KMT2AMAPK14CYP1A2
SCHEMBL13522479 0.78 MAPT (0.51) KMT2AMEN1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020022794-A1 1,3,4-OXADIAZOLE DERIVATIVE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2020-01-30 WO disclosed