SCHEMBL2648798

SCHEMBL2648798

CC(=O)Nc1cccc(-c2cnc(N(C)C)nc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 4/20 0.54
CHEK1 O14757 2/20 0.54
USP7 Q93009 1/20 0.54
FGFR1 P11362 1/20 0.54
NEK2 P51955 1/20 0.54
MAPK15 Q8TD08 1/20 0.54
NPC1 O15118 2/20 0.53
RAB9A P51151 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
TP53 P04637 1/20 0.53
STAT1 P42224 1/20 0.53
CHEK2 O96017 1/20 0.52
NQO2 P16083 2/20 0.50
NTRK1 P04629 1/20 0.50
MAP4K4 O95819 1/20 0.50
CYP17A1 P05093 1/20 0.50
CYP11B1 P15538 1/20 0.50
CYP11B2 P19099 1/20 0.50
TSHR P16473 1/20 0.50
PIP4K2A P48426 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2646435 0.79 CNR1 (0.63) FYNCHEK1USP7FGFR1NEK2
SCHEMBL11232425 0.78 FYN (0.58) FYNCHEK1USP7FGFR1NEK2
SCHEMBL3786463 0.76 NQO2 (0.73) NPC1RAB9ASMN1; SMN2TP53NQO2
SCHEMBL8577619 0.75 SMN1; SMN2 (0.70) NPC1RAB9ASMN1; SMN2TP53NQO2
SCHEMBL11222723 0.75 CNR1 (0.64) FYNNPC1RAB9ASMN1; SMN2TP53
SCHEMBL10663620 0.74 CYP17A1 (0.76) FYNNPC1RAB9ASMN1; SMN2NQO2
SCHEMBL3242870 0.74 BRAF (0.62) FYNCHEK1USP7FGFR1NEK2
SCHEMBL12821681 0.74 CHEK1 (0.69) FYNCHEK1USP7FGFR1NEK2
SCHEMBL11227834 0.74 CYP17A1 (0.56) CHEK1FGFR1NEK2MAPK15NPC1
SCHEMBL13680541 0.73 HSD17B10 (0.79) NPC1RAB9ASMN1; SMN2NQO2CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5902813-A MODULATORS OF THE BENZODIAXEPINE RECEPTOR OT THE GAMMA-BUTYRIC ACID(A) RECEPTOR COMPLEX; ANXIOLYTIC, ANTIEPILEPTIC AND -CONVULSANT AGENTS; SLEEP AND MEMORY DISORDERS NEUROSEARCH A/S (DK) 1999-05-11 US disclosed
EP-0821683-A1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABA A? RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 1998-02-04 EP disclosed
WO-1996033192-A1 BENZIMIDAZOLE COMPOUNDS AND THEIR USE AS MODULATORS OF THE GABAA RECEPTOR COMPLEX NEUROSEARCH A/S (DK) 1996-10-24 WO disclosed