SCHEMBL8577619

SCHEMBL8577619

CC(=O)Nc1ccc(-c2cccc(NC(C)=O)c2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.70
HTT P42858 1/20 0.70
L3MBTL1 Q9Y468 1/20 0.70
CYP17A1 P05093 1/20 0.64
CYP11B1 P15538 1/20 0.64
CYP11B2 P19099 1/20 0.64
HSD17B1 P14061 1/20 0.63
HSD17B2 P37059 1/20 0.63
CNR1 P21554 3/20 0.63
PIP4K2A P48426 1/20 0.62
PIP4K2B P78356 1/20 0.62
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
NQO2 P16083 2/20 0.61
ALDH1A1 P00352 3/20 0.59
HSD17B10 Q99714 2/20 0.59
MGLL Q99685 1/20 0.59
CYP1A2 P05177 1/20 0.59
NAPRT Q6XQN6 1/20 0.59
TP53 P04637 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23576901 0.91 HTT (0.63) SMN1; SMN2HTTL3MBTL1CYP17A1CYP11B1
SCHEMBL3786463 0.91 NQO2 (0.73) SMN1; SMN2CYP17A1CYP11B1CYP11B2HSD17B1
SCHEMBL12999591 0.89 NPC1 (0.69) SMN1; SMN2HTTL3MBTL1CYP17A1CYP11B1
SCHEMBL4654909 0.88 ALDH1A1 (0.67) SMN1; SMN2HTTL3MBTL1CYP17A1CYP11B1
SCHEMBL14384612 0.88 CNR1 (0.71) SMN1; SMN2CYP17A1CYP11B1CYP11B2HSD17B1
SCHEMBL969807 0.88 RAB9A (0.65) SMN1; SMN2HTTL3MBTL1CYP17A1CYP11B1
SCHEMBL1749196 0.86 MEN1 (0.59) SMN1; SMN2CYP17A1CYP11B1CYP11B2HSD17B1
SCHEMBL8265472 0.86 HSD17B10 (0.66) SMN1; SMN2HTTL3MBTL1HSD17B1HSD17B2
SCHEMBL12919978 0.85 CYP17A1 (0.60) CYP17A1CYP11B1CYP11B2HSD17B1HSD17B2
SCHEMBL6792137 0.85 CYP17A1 (0.60) SMN1; SMN2HTTL3MBTL1CYP17A1CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998014501-A1 PROCESS FOR THE PREPARATION OF THERMOTROPIC AROMATIC POLYESTERS DIRECTLY FROM DIALKYL AROMATIC ESTERS HOECHST CELANESE CORPORATION (US) 1998-04-09 WO claimed
US-5731401-A ONE STEP; HIGH MOLECULAR WEIGHT HOECHST CELANESE CORP. (US) 1998-03-24 US claimed
WO-1998014501-A1 PROCESS FOR THE PREPARATION OF THERMOTROPIC AROMATIC POLYESTERS DIRECTLY FROM DIALKYL AROMATIC ESTERS HOECHST CELANESE CORPORATION (US) 1998-04-09 WO disclosed
US-5731401-A ONE STEP; HIGH MOLECULAR WEIGHT HOECHST CELANESE CORP. (US) 1998-03-24 US disclosed