SCHEMBL2649965

SCHEMBL2649965

CC(=O)Cl.COC(=O)c1cnccn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.52
KDM4E B2RXH2 3/20 0.50
NAPRT Q6XQN6 1/20 0.50
HCAR2 Q8TDS4 1/20 0.50
SMN1; SMN2 Q16637 5/20 0.49
ALDH1A1 P00352 1/20 0.49
GAA P10253 1/20 0.49
TSHR P16473 3/20 0.48
ADORA3 P0DMS8 1/20 0.48
MC4R P32245 1/20 0.48
ADRA1A P35348 1/20 0.48
MC3R P41968 1/20 0.48
NPC1 O15118 5/20 0.48
MAPT P10636 2/20 0.46
HTT P42858 1/20 0.46
POLB P06746 3/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
USP2 O75604 1/20 0.46
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29651938 0.93 KDM4E (0.57) RAB9AKDM4ENAPRTHCAR2SMN1; SMN2
SCHEMBL108950 0.93 KDM4E (0.57) RAB9AKDM4ENAPRTHCAR2SMN1; SMN2
Hydrochloric Acid SCHEMBL29070148 0.91 KDM4E (0.55) RAB9AKDM4ENAPRTHCAR2SMN1; SMN2
Hydrochloric Acid SCHEMBL27902568 0.91 KDM4E (0.55) RAB9AKDM4ENAPRTHCAR2SMN1; SMN2
Hydrochloric Acid SCHEMBL30529579 0.91 KDM4E (0.55) RAB9AKDM4ENAPRTHCAR2SMN1; SMN2
Trifluoroacetic Acid SCHEMBL31010384 0.81 KDM4E (0.50) RAB9AKDM4ENAPRTHCAR2SMN1; SMN2
Dimethylamine SCHEMBL4392114 0.79 KDM4E (0.50) RAB9AKDM4ENAPRTHCAR2SMN1; SMN2
SCHEMBL16328267 0.78 KDM4E (0.53) RAB9AKDM4ENAPRTHCAR2SMN1; SMN2
SCHEMBL1505691 0.77 KDM4E (0.57) RAB9AKDM4ENAPRTHCAR2GAA
SCHEMBL875263 0.77 KDM4E (0.61) KDM4ENAPRTHCAR2SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1107967-A2 TRIAZOLOPYRIDAZINE DERIVATIVES FOR TREATING ANXIETY AND ENHANCING COGNITION MERCK SHARP & DOHME LTD. (GB) 2001-06-20 EP disclosed
WO-2000012505-A2 TRIAZOLOPYRIDAZINE DERIVATIVES FOR TREATING ANXIETY AND ENHANCING COGNITION MERCK SHARP & DOHME LIMITED (GB) 2000-03-09 WO disclosed