SCHEMBL26501430

SCHEMBL26501430

CC(C)(C)c1cc(N)cc(Cl)c1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.38
ALDH1A1 P00352 1/20 0.38
NR1H4 Q96RI1 3/20 0.37
THRB P10828 1/20 0.35
TSHR P16473 2/20 0.35
GLA P06280 1/20 0.35
POLB P06746 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.33
ADRB2 P07550 2/20 0.31
ADRB1 P08588 1/20 0.31
HSD11B1 P28845 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24616502 0.86 TSHR (0.43) CYP3A4ALDH1A1THRBTSHRGLA
SCHEMBL25014091 0.81 CYP3A4 (0.50) CYP3A4ALDH1A1THRBTSHRGLA
Hydrochloric Acid SCHEMBL25373977 0.79 CYP3A4 (0.48) CYP3A4ALDH1A1THRBTSHRGLA
SCHEMBL25165270 0.78 POLB (0.36) CYP3A4ALDH1A1TSHRGLAPOLB
SCHEMBL29295830 0.77 ALOX15 (0.39) CYP3A4ALDH1A1POLBMAPTCA1
SCHEMBL23206103 0.76 CYP3A4 (0.43) CYP3A4ALDH1A1THRBTSHRMAPT
SCHEMBL29676064 0.72 CYP3A4 (0.41) CYP3A4ALDH1A1THRBTSHRGAA
SCHEMBL21718397 0.72 CYP3A4 (0.41) CYP3A4ALDH1A1NR1H4THRBTSHR
SCHEMBL25417114 0.72 CYP3A4 (0.41) CYP3A4ALDH1A1THRBTSHRGAA
SCHEMBL30789287 0.72 THRB (0.39) CYP3A4ALDH1A1THRBTSHRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230321253-A1 BIFUNCTIONAL COMPOUNDS AND PHARMACEUTICAL USES THEREOF Risen (Suzhou) Pharma Tech Co., Ltd. (CN) 2023-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230321253-A1 BIFUNCTIONAL COMPOUNDS AND PHARMACEUTICAL USES THEREOF KRAS, MDM2, NRAS CYP3A4 4444/4885ALDH1A1 3243/4885NR1H4 1763/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.