SCHEMBL2651279

SCHEMBL2651279

N#Cc1cccc(NC(=O)NC(c2ccc(C(=O)NCCC(=O)O)cc2)c2ccc(C3CCCCC3)cc2)c1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GCGR P47871 5/20 0.48
EPHX2 P34913 2/20 0.44
TSHR P16473 1/20 0.43
ROCK2 O75116 3/20 0.43
KMT2A Q03164 1/20 0.42
CYP2D6 P10635 1/20 0.41
MCHR1 Q99705 1/20 0.41
CCR3 P51677 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GIPR P48546 1/20 0.39
HTR2A P28223 2/20 0.39
MAPK14 Q16539 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7101508 0.91 GCGR (0.45) GCGREPHX2TSHRROCK2MCHR1
SCHEMBL2652649 0.87 GCGR (0.50) GCGREPHX2KMT2ACYP2D6GIPR
SCHEMBL2650399 0.87 GCGR (0.50) GCGREPHX2TSHRKMT2ACYP2D6
SCHEMBL2652582 0.87 GCGR (0.51) GCGREPHX2KMT2ACYP2D6L3MBTL1
SCHEMBL6750387 0.87 GCGR (0.50) GCGREPHX2CYP2D6GIPR
SCHEMBL2651718 0.87 GCGR (0.50) GCGREPHX2CYP2D6GIPR
SCHEMBL2653146 0.87 GCGR (0.50) GCGREPHX2KMT2ACYP2D6GIPR
SCHEMBL2651202 0.87 GCGR (0.44) GCGREPHX2GIPR
SCHEMBL2658771 0.86 GCGR (0.53) GCGREPHX2CYP2D6GIPR
SCHEMBL2652856 0.85 S1PR3 (0.45) GCGREPHX2CYP2D6GIPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040127560-A1 Glucagon antagonists/inverse agonists MADSEN PETER (DK) 2004-07-01 US claimed
US-6706744-B2 HYPOGLYCEMIC AGENTS; ANTIDIABETIC AGENTS NOVO NORDISK A/S (DK) 2004-03-16 US claimed
WO-2002040444-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2002-05-23 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127560-A1 Glucagon antagonists/inverse agonists GLP1R, GPR119, GCGR GCGR 3/4885EPHX2 2973/4885TSHR 78/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.