SCHEMBL2651960

SCHEMBL2651960

N#Cc1cccc(-c2cccc(N)c2)c1F

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.44
MAP4K4 O95819 2/20 0.44
MAOA P21397 1/20 0.41
ALOX5AP P20292 1/20 0.40
FEN1 P39748 1/20 0.40
ADORA2A P29274 1/20 0.40
USP30 Q70CQ3 2/20 0.38
CYP11B2 P19099 2/20 0.38
CYP11B1 P15538 1/20 0.38
NTRK1 P04629 2/20 0.38
LRRK2 Q5S007 2/20 0.38
PIK3CA P42336 1/20 0.38
MECP2 P51608 1/20 0.37
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
AR P10275 1/20 0.36
BACE1 P56817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL979345 0.84 IKBKB (0.50) IKBKBMAP4K4MAOAALOX5APFEN1
SCHEMBL31006072 0.81 IKBKB (0.51) IKBKBMAP4K4MAOAADORA2ANTRK1
SCHEMBL4975197 0.80 ESR2 (0.48) MAOACYP11B2CYP11B1LRRK2AR
SCHEMBL2649762 0.79 GRM5 (0.41) IKBKBMAP4K4MAOAALOX5APFEN1
SCHEMBL22211410 0.78 CTSS (0.49) CYP11B2CYP11B1AR
SCHEMBL12679951 0.77 IKBKB (0.56) IKBKBMAP4K4MAOAADORA2ANTRK1
SCHEMBL3786949 0.77 MAP4K4 (0.50) MAP4K4MAOAMECP2
SCHEMBL12707386 0.77 MAOA (0.41) IKBKBMAP4K4MAOAALOX5APFEN1
SCHEMBL28662059 0.75 CA1 (0.45) ALOX5APFEN1ADORA2AUSP30CYP11B2
SCHEMBL980699 0.75 CYP11B1 (0.49) MAP4K4MAOACYP11B2CYP11B1PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381606-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2004-01-21 EP disclosed
WO-2002074773-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-09-26 WO disclosed