SCHEMBL26546263

SCHEMBL26546263

COc1cccc(CNc2ccc(SNc3cccc(N4CCNCC4)c3)cc2)c1O

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX12 P18054 12/20 0.70
MAPT P10636 5/20 0.45
GAA P10253 3/20 0.45
CCNE1 P24864 1/20 0.44
CDK2 P24941 1/20 0.44
ALOX15 P16050 4/20 0.44
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPK1 P28482 3/20 0.44
TDP1 Q9NUW8 3/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
NPSR1 Q6W5P4 2/20 0.44
HTT P42858 2/20 0.44
MEN1 O00255 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
NPC1 O15118 1/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26546267 0.92 ALOX12 (0.68) ALOX12MAPTGAACCNE1CDK2
SCHEMBL26546300 0.85 ALOX12 (0.70) ALOX12MAPTGAACCNE1CDK2
SCHEMBL16646181 0.82 ALOX12 (1.00) ALOX12ALOX15
SCHEMBL30580748 0.82 ALOX12 (1.00) ALOX12ALOX15
SCHEMBL26546404 0.82 ALOX12 (0.70) ALOX12MAPTGAAALOX15KDM4E
SCHEMBL26546259 0.79 ALOX12 (0.66) ALOX12MAPTGAAALOX15KDM4E
SCHEMBL30580749 0.75 ALOX12 (1.00) ALOX12ALOX15
SCHEMBL16646068 0.75 ALOX12 (1.00) ALOX12ALOX15
SCHEMBL26546320 0.75 ALOX12 (0.66) ALOX12MAPTGAAALOX15KDM4E
SCHEMBL26546203 0.72 KDM4E (0.77) ALOX12MAPTGAAALOX15KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3054936-B1 4-((2-HYDROXY-3-METHOXYBENZYL)AMINO) BENZENESULFONAMIDE DERIVATIVES AS 12-LIPOXYGENASE INHIBITORS EASTERN VIRGINIA MEDICAL SCHOOL (US) 2023-10-18 EP disclosed