SCHEMBL26547288

SCHEMBL26547288

CC(C)(C)N1CCCNc2ncccc21

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
GFER P55789 1/20 0.37
KMT2A Q03164 1/20 0.37
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
SLC6A4 P31645 1/20 0.35
EPHX2 P34913 1/20 0.34
AKT1 P31749 2/20 0.33
HTR1A P08908 1/20 0.32
SLC6A2 P23975 1/20 0.32
HTR7 P34969 1/20 0.31
IDH1 O75874 2/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRL1 P41146 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
CHRNB2 P17787 1/20 0.30
CHRNA4 P43681 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25094286 0.90 HTR2A (0.36) HTR2AHTR2CSLC6A4EPHX2AKT1
SCHEMBL26547286 0.76 BRD4 (0.39) MEN1RAB9AGFERKMT2AHTR1A
SCHEMBL26547290 0.75 EPHX2 (0.37) MEN1RAB9AGFERKMT2AHTR2A
SCHEMBL10222503 0.74 KCNQ2 (0.40) MEN1KMT2A
SCHEMBL25646141 0.74 OPRM1 (0.40) MEN1KMT2AAKT1IDH1OPRM1
SCHEMBL19754379 0.73 KCNQ2 (0.44) MEN1KMT2A
SCHEMBL517896 0.71 HTR2A (0.42) MEN1RAB9AGFERKMT2AHTR2A
SCHEMBL14279926 0.70 KCNQ2 (0.36) HTR2AHTR2CSLC6A4EPHX2
SCHEMBL23344744 0.69 GAA (0.41) HTR2AEPHX2HTR1AHTR7
SCHEMBL24635835 0.68 HTR2A (0.36) HTR2AHTR2CSLC6A4EPHX2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230322724-A1 HETEROCYCLIC COMPOUNDS AS CBP/EP300 BROMODOMAIN INHIBITORS AURIGENE ONCOLOGY LIMITED (IN) 2023-10-12 US disclosed
US-20230322724-A1 HETEROCYCLIC COMPOUNDS AS CBP/EP300 BROMODOMAIN INHIBITORS AURIGENE ONCOLOGY LIMITED (IN) 2023-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230322724-A1 HETEROCYCLIC COMPOUNDS AS CBP/EP300 BROMODOMAIN INHIBITORS EP300, HDAC1, BRD3 MEN1 2797/4885RAB9A 3660/4885GFER 4368/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.