SCHEMBL26547290

SCHEMBL26547290

CC(C)(C)N1CCCNc2cccnc21

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.37
MEN1 O00255 1/20 0.34
RAB9A P51151 1/20 0.34
GFER P55789 1/20 0.34
KMT2A Q03164 1/20 0.34
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
CNR2 P34972 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26547297 0.90 EPHX2 (0.39) EPHX2HTR2AHTR2CHTR2BGAA
SCHEMBL7017304 0.79 MEN1 (0.50) EPHX2MEN1RAB9AGFERKMT2A
SCHEMBL26547286 0.76 BRD4 (0.39) MEN1RAB9AGFERKMT2AGAA
SCHEMBL26547288 0.75 MEN1 (0.37) EPHX2MEN1RAB9AGFERKMT2A
SCHEMBL6980295 0.74 HDAC6 (0.40) KMT2AHTR2AHTR2CHTR2B
SCHEMBL19754380 0.73 HDAC6 (0.40) KMT2AHTR2AHTR2CHTR2BCYP1A2
SCHEMBL12405333 0.71 MEN1 (0.38) EPHX2MEN1RAB9AGFERKMT2A
SCHEMBL12049049 0.70 MTNR1A (0.43) EPHX2HTR2AHTR2CHTR2BCYP1A2
SCHEMBL11584126 0.70 EPHX2 (0.41) EPHX2GAA
SCHEMBL26549764 0.70 CYP2D6 (0.37) MEN1KMT2ACYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230322724-A1 HETEROCYCLIC COMPOUNDS AS CBP/EP300 BROMODOMAIN INHIBITORS AURIGENE ONCOLOGY LIMITED (IN) 2023-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230322724-A1 HETEROCYCLIC COMPOUNDS AS CBP/EP300 BROMODOMAIN INHIBITORS EP300, HDAC1, BRD3 EPHX2 1846/4885MEN1 2797/4885RAB9A 3660/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.