SCHEMBL265486

SCHEMBL265486

OCc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.52
RXRA P19793 2/20 0.51
RXRB P28702 2/20 0.51
RXRG P48443 2/20 0.51
CES2 O00748 1/20 0.46
PRKCA P17252 1/20 0.45
PRKCD Q05655 1/20 0.45
ACHE P22303 1/20 0.42
MTOR P42345 1/20 0.41
DAO P14920 2/20 0.40
TACR1 P25103 4/20 0.40
MLYCD O95822 1/20 0.40
ACP3 P15309 1/20 0.38
KIF11 P52732 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12871778 0.89 RXRA (0.45) IDO1RXRARXRBRXRGCES2
SCHEMBL3279035 0.86 RXRA (0.46) IDO1RXRARXRBRXRGCES2
SCHEMBL29876769 0.86 RXRA (0.46) IDO1RXRARXRBRXRGCES2
SCHEMBL21474429 0.86 ACHE (0.58) IDO1RXRARXRBRXRGCES2
SCHEMBL16951240 0.84 RXRA (0.45) IDO1RXRARXRBRXRGCES2
SCHEMBL799344 0.84 RXRA (0.45) IDO1RXRARXRBRXRGPRKCA
SCHEMBL2773850 0.84 RXRA (0.45) IDO1RXRARXRBRXRGCES2
SCHEMBL630541 0.84 RXRA (0.45) IDO1RXRARXRBRXRGPRKCA
SCHEMBL129085 0.84 RXRA (0.45) IDO1RXRARXRBRXRGCES2
SCHEMBL130263 0.84 RXRA (0.45) IDO1RXRARXRBRXRGCES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 557 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113999342-B Migratable polymer-based functional modifier and preparation method and application thereof 厦门大学 2022-08-12 CN claimed
CN-113999342-A Migratable polymer-based functional modifier and preparation method and application thereof 厦门大学 2022-02-01 CN claimed
CN-113214045-A Preparation process of high-purity 3, 5-bis (trifluoromethyl) benzyl alcohol 宁夏忠同生物科技有限公司 2021-08-06 CN claimed
US-9616459-B1 Polymeric coatings for fortification of visible, infrared, and laser optical devices LOCKHEED MARTIN CORPORATION (US) 2017-04-11 US claimed
US-8952083-B2 Fluorocopolymer composition and its production process ASAHI GLASS COMPANY, LIMITED (JP) 2015-02-10 US claimed
EP-1993991-B1 PROCESS FOR THE PREPARATION OF 3,5-BIS (TRIFLUOROMETHYL)-N-METHYLBENZYLAMINE MITENI SPA (IT) 2010-09-22 EP claimed
EP-1993991-A2 PROCESS FOR THE PREPARATION OF 3,5-BIS (TRIFLUOROMETHYL)-N-METHYLBENZYLAMINE MITENI S.p.A. (IT) 2008-11-26 EP claimed
EP-1115693-B9 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL $i(TERTIARY)-HETEROALKYLAMINES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY MONSANTO CO (US) 2007-12-19 EP claimed
WO-2007107818-A2 PROCESS FOR THE PREPARATION OF 3,5-BIS (TRIFLUOROMETHYL)-N-METHYLBENZYLAMINE MITENI S.P.A. (IT) 2007-09-27 WO claimed
EP-1673329-B1 PROCESS FOR THE PREPARATION 3,5-BIS(TRIFLUOROMETHYL)BENZYLALCOHOL MITENI SPA (IT) 2007-09-12 EP claimed
EP-1115695-A1 (R)-CHIRAL HALOGENATED 1-SUBSTITUTEDAMINO-(N+1)-ALKANOLS USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY Monsanto Company (US) 2001-07-18 EP claimed
EP-1115693-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL $i(TERTIARY)-HETEROALKYLAMINES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY Monsanto Company (US) 2001-07-18 EP claimed
EP-1115694-A1 SUBSTITUTED N-ALIPHATIC-N-AROMATIC (TERTIARY)-HETEROALKYLAMINES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY Monsanto Company (US) 2001-07-18 EP claimed
WO-2000018724-A1 (R)-CHIRAL HALOGENATED 1-SUBSTITUTEDAMINO-(n+1)-ALKANOLS USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY MONSANTO COMPANY (US) 2000-04-06 WO claimed
WO-2000018723-A1 SUBSTITUTED N-ALIPHATIC-N-AROMATIC TERTIARY-HETEROALKYLAMINES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY MONSANTO COMPANY (US) 2000-04-06 WO claimed
WO-2000018721-A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL TERTIARY-HETEROALKYLAMINES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY MONSANTO COMPANY (US) 2000-04-06 WO claimed
US-5922117-A Ink compositions containing alcohols XEROX CORPORATION (US) 1999-07-13 US claimed
US-5897940-A Ink jet transparencies XEROX CORPORATION (US) 1999-04-27 US claimed
US-5663265-A FREE RADICAL COPOLYMERIZATION FOR COATINGS HOECHST AKTIENGESELLSCHAFT (DE) 1997-09-02 US claimed
US-5596057-A INTERPOLYMER FROM STERICALLY HINDERED UNSATURATED ESTERS HOECHST AKTIENGESELLSCHAFT (DE) 1997-01-21 US claimed