SCHEMBL265949

SCHEMBL265949

NC1CCc2ccc(O)cc2C1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 9/20 1.00
DRD3 P35462 9/20 1.00
OPRK1 P41145 1/20 0.86
MAPT P10636 2/20 0.63
NFKB1 P19838 1/20 0.63
THPO P40225 1/20 0.63
HIF1A Q16665 1/20 0.63
HSD17B10 Q99714 1/20 0.63
USP2 O75604 1/20 0.63
ALDH1A1 P00352 1/20 0.63
KDM4E B2RXH2 1/20 0.61
DRD4 P21917 6/20 0.57
PLAU P00749 1/20 0.57
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HTR1A P08908 1/20 0.50
ACHE P22303 1/20 0.50
ADRB2 P07550 1/20 0.50
CYP2D6 P10635 1/20 0.50
CASP1 P29466 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30697493 1.00 DRD2 (1.00) DRD2DRD3OPRK1MAPTNFKB1
SCHEMBL5722322 1.00 DRD2 (1.00) DRD2DRD3OPRK1MAPTNFKB1
SCHEMBL9135070 1.00 DRD2 (1.00) DRD2DRD3OPRK1MAPTNFKB1
SCHEMBL30839518 1.00 DRD2 (1.00) DRD2DRD3OPRK1MAPTNFKB1
Bromide SCHEMBL354391 0.98 DRD2 (0.96) DRD2DRD3OPRK1MAPTNFKB1
Hydrochloric Acid SCHEMBL9317222 0.98 DRD2 (0.96) DRD2DRD3OPRK1MAPTNFKB1
Water SCHEMBL9305270 0.98 DRD2 (0.96) DRD2DRD3OPRK1MAPTNFKB1
Water SCHEMBL9305264 0.98 DRD2 (0.96) DRD2DRD3OPRK1MAPTNFKB1
Bromide SCHEMBL5722309 0.98 DRD2 (0.96) DRD2DRD3OPRK1MAPTNFKB1
Bromide SCHEMBL354286 0.98 DRD2 (0.96) DRD2DRD3OPRK1MAPTNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 109 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108455563-A A kind of preparation method of Nitrogen-rich porous carbon microballoon 天津工业大学 2018-08-28 CN claimed
EP-0347313-B1 2-Amino-7-hydroxytetraline ethers SANOFI ELF (FR) 1993-12-15 EP claimed
EP-0383686-B1 2-AMINO-7-HYDROXYTETRALINE CARBOXYALKYL ETHERS ELF SANOFI (FR) 1993-08-04 EP claimed
US-5202466-A 2-amino-7-hydroxytetraline ethers SANOFI (FR) 1993-04-13 US claimed
US-5198586-A Process for the preparation of phenylethanolaminotetralins SANOFI (FR) 1993-03-30 US claimed
US-5159103-A 2-amino-7-hydroxytetraline ethers SANOFI (FR) 1992-10-27 US claimed
EP-0303545-B1 PROCESS FOR THE PREPARATION OF PHENYLETHANOLAMINOTETRALINES ELF SANOFI (FR) 1992-06-17 EP claimed
EP-0383686-A1 2-Amino-7-hydroxytetraline carboxyalkyl ethers ELF SANOFI (FR) 1990-08-22 EP claimed
EP-0347313-A2 2-Amino-7-hydroxytetraline ethers ELF SANOFI (FR) 1989-12-20 EP claimed
EP-0303545-A2 Process for the preparation of phenylethanolaminotetralines ELF SANOFI (FR) 1989-02-15 EP claimed
JP-2196760-A None JP disclosed
US-11970512-B2 Amphotericin B derivatives with improved therapeutic index THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2024-04-30 US disclosed
CN-110407898-B Amphotericin B derivatives with improved therapeutic index 伊利诺伊大学评议会 2023-12-01 CN disclosed
CN-110831600-B Indole AHR inhibitors and uses thereof 医肯纳肿瘤学公司 2023-10-17 CN disclosed
US-20230028336-A1 INDOLE AHR INHIBITORS AND USES THEREOF PAHR THERAPEUTICS, INC. 2023-01-26 US disclosed
EP-0347313-A2 2-Amino-7-hydroxytetraline ethers ELF SANOFI (FR) 1989-12-20 EP disclosed
WO-1989009050-A1 THERAPEUTICALLY USEFUL TETRALIN DERIVATIVES THE UPJOHN COMPANY (US) 1989-10-05 WO disclosed
EP-0334538-A1 Therapeutically useful tetralin derivatives THE UPJOHN COMPANY (US) 1989-09-27 EP disclosed
EP-0303545-A2 Process for the preparation of phenylethanolaminotetralines ELF SANOFI (FR) 1989-02-15 EP disclosed
EP-0303545-A2 Process for the preparation of phenylethanolaminotetralines ELF SANOFI (FR) 1989-02-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230028336-A1 INDOLE AHR INHIBITORS AND USES THEREOF AHR, ARNT, IDO1 DRD2 1634/4885DRD3 1688/4885OPRK1 176/4885
US-11970512-B2 Amphotericin B derivatives with improved therapeutic index C9, AMPD3, C5 DRD2 4145/4885DRD3 2361/4885OPRK1 4776/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.