SCHEMBL2659900

SCHEMBL2659900

Clc1cc(Br)ccc1-c1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 6/20 0.54
CYP11B2 P19099 6/20 0.54
CYP2A6 P11509 5/20 0.50
KMT2A Q03164 2/20 0.49
KDM4E B2RXH2 1/20 0.49
MEN1 O00255 1/20 0.49
MAPK1 P28482 1/20 0.49
HTT P42858 1/20 0.49
CYP17A1 P05093 4/20 0.48
CYP3A4 P08684 3/20 0.48
ALDH1A1 P00352 1/20 0.47
CYP1A2 P05177 1/20 0.47
MKNK1 Q9BUB5 1/20 0.44
MKNK2 Q9HBH9 1/20 0.44
RXFP1 Q9HBX9 2/20 0.44
CYP19A1 P11511 2/20 0.43
PRNP P04156 1/20 0.43
PPARG P37231 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
NR2E3 Q9Y5X4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2652392 0.86 CYP11B1 (0.54) CYP11B1CYP11B2CYP2A6KMT2AKDM4E
SCHEMBL28300994 0.84 CYP11B1 (0.59) CYP11B1CYP11B2CYP2A6KMT2AKDM4E
SCHEMBL2659447 0.79 CYP11B1 (0.54) CYP11B1CYP11B2CYP2A6KMT2ACYP17A1
SCHEMBL19257504 0.79 CYP11B1 (0.54) CYP11B1CYP11B2CYP2A6KMT2AKDM4E
SCHEMBL21588612 0.79 CYP11B1 (0.54) CYP11B1CYP11B2CYP2A6KMT2AKDM4E
SCHEMBL21044098 0.79 AXL (0.56) CYP11B1CYP11B2CYP2A6KDM4EMEN1
SCHEMBL2402017 0.77 CYP2A6 (0.54) CYP2A6MAPK1ALDH1A1CYP19A1NPSR1
SCHEMBL2649040 0.76 CYP11B2 (0.54) CYP11B1CYP11B2CYP2A6KMT2AMAPK1
SCHEMBL6222583 0.76 CYP11B1 (0.54) CYP11B1CYP11B2CYP2A6KMT2AKDM4E
SCHEMBL551165 0.76 NPC1 (0.65) CYP11B1CYP2A6KDM4EHTTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381606-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2004-01-21 EP disclosed
WO-2002074773-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-09-26 WO disclosed