SCHEMBL2661888

SCHEMBL2661888

CC(C)(O)c1ncn2c(-c3ccc(F)c(-c4c(F)cccc4C#N)c3)cnc2c1F

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 20/20 0.61
GABRG2 P18507 20/20 0.61
GABRB3 P28472 20/20 0.61
GABRA3 P34903 18/20 0.61
GABRA5 P31644 14/20 0.61
GABRA2 P47869 7/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2659993 0.89 GABRA1 (0.60) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2657350 0.88 GABRA1 (0.49) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2659106 0.86 GABRA1 (0.80) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2659942 0.86 GABRA1 (0.58) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2659826 0.81 GABRA1 (0.59) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2658248 0.80 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2658754 0.80 GABRG2 (0.62) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2656804 0.80 GABRA1 (0.47) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL2657951 0.79 GABRA1 (0.68) GABRA1GABRG2GABRB3GABRA3GABRA5
SCHEMBL31678897 0.77 GABRA1 (0.77) GABRA1GABRG2GABRB3GABRA3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004065388-A1 FLUOROIMIDAZOPYRIMIDINES AS GABA-A ALPHA 2/3 LIGANDS FOR DEPRESSION/ANXIETY MERCK SHARP & DOHME LIMITED (GB) 2004-08-05 WO disclosed