SCHEMBL2662687

SCHEMBL2662687

O=C(Cl)C(Br)c1ccccc1F

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 5/20 0.46
CES1 P23141 5/20 0.46
ALDH1A1 P00352 1/20 0.45
ALOX15 P16050 1/20 0.45
GAA P10253 1/20 0.41
CNR2 P34972 2/20 0.40
HDAC4 P56524 3/20 0.39
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP3A4 P08684 1/20 0.35
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30888308 0.82 CES2 (0.47) CES2CES1ALDH1A1ALOX15GAA
SCHEMBL3635938 0.82 CES2 (0.47) CES2CES1ALDH1A1ALOX15GAA
SCHEMBL8127998 0.82 CES2 (0.47) CES2CES1ALDH1A1ALOX15GAA
SCHEMBL7470109 0.80 GAA (0.49) CES2CES1ALDH1A1ALOX15GAA
SCHEMBL11965195 0.80 CES2 (0.46) CES2CES1ALDH1A1ALOX15GAA
SCHEMBL7724344 0.79 CES2 (0.48) CES2CES1ALDH1A1ALOX15GAA
SCHEMBL9297918 0.78 ACP3 (0.42) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL29362410 0.78 CES2 (0.61) CES2CES1ALDH1A1ALOX15GAA
SCHEMBL9297917 0.78 ACP3 (0.42) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL1885454 0.78 CES2 (0.47) CES2CES1ALDH1A1ALOX15GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105051036-B Flavonoid or isoflavone compound and application thereof 上海正基医药科技有限公司 2017-09-29 CN disclosed
EP-1212324-B1 IMIDAZO-TRIAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME (GB) 2003-10-29 EP disclosed
US-6608062-B1 Ligands for gamma-aminobutyric acid receptors; treatment and/or prevention of central nervous system disorders, including anxiety MERCK SHARP & DOHME LTD. 2003-08-19 US disclosed
EP-1212324-A1 IMIDAZO-TRIAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LTD. (GB) 2002-06-12 EP disclosed
WO-2001014377-A1 IMIDAZO-TRIAZINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2001-03-01 WO disclosed
CN-1039713-C 3-chloroheterobicyclo [3.1.0] hexane-2-one derivatives and herbicidal compositions containing them as herbicidal active ingredients MITSUI TOATSU CHEMICALS (JP) 1998-09-09 CN disclosed
EP-0600507-B1 3-Azabicyclo(3.1.0.)hexane-2-one derivatives and Herbicidal Compositions Containing them as Herbicidally Active Ingredients MITSUI TOATSU CHEMICALS (JP) 1996-03-06 EP disclosed
US-5352655-A Pre- and postemergence; rice MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-10-04 US disclosed
EP-0600507-A1 3-Azabicyclo(3.1.0.)hexane-2-one derivatives and Herbicidal Compositions Containing them as Herbicidally Active Ingredients MITSUI TOATSU CHEMICALS, Inc. (JP) 1994-06-08 EP disclosed