SCHEMBL2665463

SCHEMBL2665463

CCN(c1ccccc1)S(=O)(=O)c1cccc(NC(=O)N(Cc2ccc(C(=O)NCC(F)C(=O)O)cc2)c2ccc(C3CCCCC3)cc2)c1

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GCGR P47871 14/20 0.60
GIPR P48546 12/20 0.60
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
STAT3 P40763 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2665459 0.92 GCGR (0.62) GCGRGIPROPRM1OPRK1MAPT
SCHEMBL2665786 0.90 GCGR (0.66) GCGRGIPROPRM1OPRK1
SCHEMBL9071759 0.90 GCGR (0.57) GCGRGIPROPRM1OPRK1STAT3
SCHEMBL2650880 0.89 GCGR (0.67) GCGRGIPROPRM1OPRK1
SCHEMBL9071304 0.88 GCGR (0.55) GCGRGIPROPRM1OPRK1STAT3
SCHEMBL2665464 0.87 GCGR (0.62) GCGRGIPRMAPT
SCHEMBL9071788 0.86 GCGR (0.68) GCGRGIPRSTAT3
SCHEMBL2665594 0.86 GCGR (0.69) GCGRGIPRSTAT3
SCHEMBL9071764 0.85 GCGR (0.69) GCGRGIPR
SCHEMBL9071761 0.84 GCGR (0.70) GCGRGIPRSTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002000612-A1 GLUCAGON ANTAGONISTS/INVERSE AGONISTS NOVO NORDISK A/S (DK) 2002-01-03 WO disclosed