SCHEMBL2666243

SCHEMBL2666243

Cc1ccnc(-c2ccc(Cl)c(F)c2)n1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KMO O15229 2/20 0.47
DYRK1A Q13627 2/20 0.43
CLK4 Q9HAZ1 2/20 0.43
GRM2 Q14416 3/20 0.40
KDM4C Q9H3R0 2/20 0.40
TRPV1 Q8NER1 1/20 0.38
EGLN2 Q96KS0 1/20 0.38
CYP1A2 P05177 1/20 0.38
ABL1 P00519 1/20 0.37
KCNH2 Q12809 1/20 0.37
GRM5 P41594 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2666270 0.87 KMO (0.47) KMODYRK1ACLK4GRM2ABL1
SCHEMBL2666251 0.85 NPC1 (0.49) KMOCLK4GRM5
SCHEMBL2666284 0.83 MEN1 (0.40) KMODYRK1ACLK4CYP1A2KCNH2
SCHEMBL22578238 0.81 CYP1A2 (0.47) KMODYRK1ACLK4CYP1A2
SCHEMBL22130225 0.81 KIT (0.41) KMO
SCHEMBL31533414 0.81 CYP17A1 (0.46)
SCHEMBL2666240 0.80 NOTUM (0.50) GRM2KDM4CCYP1A2
SCHEMBL20597708 0.77 KMO (0.44) KMODYRK1ACLK4GRM2KDM4C
SCHEMBL8226435 0.77 RXRA (0.44) DYRK1ACLK4CYP1A2
SCHEMBL12021925 0.77 MEN1 (0.34) KMODYRK1ACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728227-B1 ORGANIC MOLECULES WITH A PYRIDINE-PHENYL CORE FOR USE IN OPTOELECTRONIC DEVICES SAMSUNG DISPLAY CO LTD (KR) 2023-08-16 EP disclosed
EP-3728227-A1 ORGANIC MOLECULES WITH A PYRIDINE-PHENYL CORE FOR USE IN OPTOELECTRONIC DEVICES cynora GmbH (DE) 2020-10-28 EP disclosed
WO-2002076983-A1 IMIDAZO-PYRIMIDINE DERIVATIVES AS LIGANDS FOR GABA RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 2002-10-03 WO disclosed