SCHEMBL2669019

SCHEMBL2669019

COCCOc1cc(CC(=O)OCc2ccccc2)cc(Oc2ccc(S(C)(=O)=O)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
MAPK1 P28482 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GCK P35557 9/20 0.42
FFAR1 O14842 2/20 0.42
LMNA P02545 2/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
MITF O75030 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
CCR6 P51684 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NR3C1 P04150 1/20 0.40
FAAH O00519 1/20 0.40
KCNH2 Q12809 1/20 0.39
ALOX5 P09917 1/20 0.39
PTPN1 P18031 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1107547 0.85 GCK (0.52) ALDH1A1MAPK1GCKLMNAMEN1
SCHEMBL2669005 0.85 GCK (0.47) GCKFFAR1KCNH2
SCHEMBL1107744 0.78 GCK (0.56) GCKMEN1KMT2AKCNH2
SCHEMBL21704383 0.76 ALDH1A1 (0.70) ALDH1A1MAPK1L3MBTL1LMNAMEN1
SCHEMBL12594271 0.76 GCK (0.53) GCKKCNH2
SCHEMBL1107721 0.75 GCK (0.55) GCKMAPTKCNH2
SCHEMBL2668841 0.75 GCK (0.53) GCKKCNH2
SCHEMBL2656511 0.75 HPGD (0.52) ALDH1A1GCKFFAR1LMNAMEN1
SCHEMBL2668144 0.74 GCK (0.46) GCKMEN1NPC1MAPTRAB9A
SCHEMBL18179855 0.74 ALDH1A1 (0.69) ALDH1A1MAPK1L3MBTL1FFAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008005964-A2 PHOSPHONATE AND PHOSPHINATE COMPOUNDS AS GLUCOKINASE ACTIVATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2008-01-10 WO disclosed