SCHEMBL2669341

SCHEMBL2669341

CN/C=C\C(=N)NC(=O)c1cc(Oc2ccc(C(=O)N3CCC3)c(F)c2)c2c(c1)OC(C)(COC)C2

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GCK P35557 5/20 0.59
CPS1 P31327 3/20 0.40
GPR119 Q8TDV5 2/20 0.33
CNR1 P21554 1/20 0.31
SLC6A4 P31645 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
HPGD P15428 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2669385 0.94 GCK (0.67) GCKCPS1GPR119CNR1SLC6A4
SCHEMBL2669283 0.91 GCK (0.66) GCKCPS1GPR119CNR1SLC6A4
SCHEMBL2643543 0.85 GCK (0.62) GCKCPS1GPR119CNR1
SCHEMBL2669286 0.82 GCK (0.55) GCKCPS1GPR119
SCHEMBL642364 0.82 GCK (0.82) GCKCPS1
SCHEMBL9071945 0.82 GCK (0.55) GCKCPS1
SCHEMBL2669367 0.82 GCK (0.55) GCKCPS1
SCHEMBL643331 0.82 GCK (0.58) GCKCPS1GPR119CNR1
SCHEMBL9923383 0.82 GCK (0.53) GCKCPS1
SCHEMBL2669284 0.80 GCK (0.52) GCKCPS1CNR1SLC6A4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463283-A1 Fused phenyl Amido heterocyclic compounds for the prevention and treatment of glucokinase-mediated diseases Pfizer Products Inc. (US) 2012-06-13 EP disclosed
WO-2007122482-A1 FUSED PHENYL AMIDO HETEROCYCLIC COMPOUNDS FOR THE PREVENTION AND TREATMENT OF GLUCOKINASE-MEDIATED DISEASES PFIZER PRODUCTS INC. (US) 2007-11-01 WO disclosed