SCHEMBL2669283

SCHEMBL2669283

CN/C=C\C(=N)NC(=O)c1cc(Oc2ccc(C(=O)N3CCC3)c(F)c2)c2c(c1)OC(C)(C)C2

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GCK P35557 5/20 0.66
CPS1 P31327 4/20 0.42
SLC6A4 P31645 3/20 0.32
HRH3 Q9Y5N1 3/20 0.32
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
GPR119 Q8TDV5 2/20 0.32
CNR1 P21554 3/20 0.31
EZH2 Q15910 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2669385 0.91 GCK (0.67) GCKCPS1SLC6A4HRH3GPR119
SCHEMBL2669286 0.91 GCK (0.55) GCKCPS1GPR119
SCHEMBL9071945 0.91 GCK (0.55) GCKCPS1
SCHEMBL2669341 0.91 GCK (0.59) GCKCPS1SLC6A4HRH3GPR119
SCHEMBL2669367 0.91 GCK (0.55) GCKCPS1EZH2
SCHEMBL9923383 0.89 GCK (0.53) GCKCPS1SCN9A
SCHEMBL2669284 0.89 GCK (0.52) GCKCPS1SLC6A4HRH3CNR1
SCHEMBL9071966 0.89 GCK (0.53) GCKEZH2
SCHEMBL2669236 0.87 GCK (0.49) GCKEZH2
SCHEMBL2669401 0.87 GCK (0.52) GCKHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463283-A1 Fused phenyl Amido heterocyclic compounds for the prevention and treatment of glucokinase-mediated diseases Pfizer Products Inc. (US) 2012-06-13 EP disclosed
WO-2007122482-A1 FUSED PHENYL AMIDO HETEROCYCLIC COMPOUNDS FOR THE PREVENTION AND TREATMENT OF GLUCOKINASE-MEDIATED DISEASES PFIZER PRODUCTS INC. (US) 2007-11-01 WO disclosed