SCHEMBL2669401

SCHEMBL2669401

CN/C=C\C(=N)NC(=O)c1cc(Oc2cnc(C(=O)N3CCC3)c(F)c2)c2c(c1)OC(C)(C)C2

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GCK P35557 12/20 0.52
GPR183 P32249 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9071971 0.90 GCK (0.42) GCK
SCHEMBL2669314 0.87 GCK (0.40) GCK
SCHEMBL2669283 0.87 GCK (0.66) GCKHRH3
SCHEMBL9071954 0.86 GCK (0.48) GCKGPR183HRH3
SCHEMBL2643740 0.84 GCK (0.54) GCKHRH3
SCHEMBL2669282 0.84 GCK (0.49) GCKHRH3
SCHEMBL2669284 0.81 GCK (0.52) GCKHRH3
SCHEMBL12101378 0.81 GCK (0.51) GCKGPR183HRH3
SCHEMBL644094 0.80 GCK (0.79) GCK
SCHEMBL15780551 0.79 GCK (0.42) GCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007122482-A1 FUSED PHENYL AMIDO HETEROCYCLIC COMPOUNDS FOR THE PREVENTION AND TREATMENT OF GLUCOKINASE-MEDIATED DISEASES PFIZER PRODUCTS INC. (US) 2007-11-01 WO disclosed