SCHEMBL26698277

SCHEMBL26698277

CN1CCC(C(C(N)=O)c2ccccc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 4/20 0.58
CACNA2D1 P54289 4/20 0.50
CACNA1B Q00975 4/20 0.50
CACNB1 Q02641 4/20 0.50
CACNA1C Q13936 4/20 0.50
CHRM2 P08172 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
CYP2D6 P10635 1/20 0.47
CHRM1 P11229 1/20 0.47
DRD1 P21728 1/20 0.47
SLC6A2 P23975 1/20 0.47
ADRA1A P35348 1/20 0.47
OPRM1 P35372 1/20 0.47
DRD3 P35462 1/20 0.47
SLC6A3 Q01959 1/20 0.47
KCNH2 Q12809 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
KDM4E B2RXH2 1/20 0.47
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26698301 0.87 CHRM3 (0.61) CHRM3CACNA2D1CACNA1BCACNB1CACNA1C
SCHEMBL4176732 0.86 HTR1E (0.51) CHRM3MEN1KMT2ALMNAMAPT
SCHEMBL22188704 0.86 HTR1E (0.51) CHRM3MEN1KMT2ALMNAMAPT
SCHEMBL6988817 0.84 HRH3 (0.49) CHRM3CYP2D6CHRM1KCNH2HRH3
SCHEMBL4866289 0.83 HTR1E (0.61) CHRM3CHRM2HTR1AADRA2ACYP2D6
SCHEMBL5049598 0.83 HTR1E (0.57) CHRM3CHRM2HTR1AADRA2ACYP2D6
SCHEMBL15797674 0.83 CHRM1 (0.44) CHRM3CHRM1KCNH2KDM4ELMNA
Hydrochloric Acid SCHEMBL5051899 0.81 HTR1E (0.59) CHRM3CHRM2HTR1AADRA2ACYP2D6
SCHEMBL5051927 0.81 MEN1 (0.59) CHRM3CHRM2HTR1AADRA2ACYP2D6
SCHEMBL14453324 0.81 MEN1 (0.59) CHRM3CHRM2HTR1AADRA2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023226965-A1 ROCK INHIBITORS AND USES THEREOF DIZAL (JIANGSU) PHARMACEUTICAL CO., LTD. (CN) 2023-11-30 WO disclosed