Clobenzorex

Clobenzorex

SCHEMBL26720

CC(Cc1ccccc1)NCc1ccccc1Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 1.00
SIGMAR1 Q99720 12/20 0.66
POLB P06746 1/20 0.65
MAPK1 P28482 1/20 0.65
CYP1A2 P05177 1/20 0.56
CYP3A4 P08684 1/20 0.56
CYP2D6 P10635 1/20 0.56
TSHR P16473 1/20 0.56
ATM Q13315 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
TAAR1 Q96RJ0 2/20 0.50
SLC18A2 Q05940 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clobenzorex SCHEMBL31080692 1.00 LMNA (1.00) LMNASIGMAR1POLBMAPK1CYP1A2
Clobenzorex SCHEMBL1649957 0.97 LMNA (0.94) LMNASIGMAR1POLBMAPK1CYP1A2
Clobenzorex SCHEMBL13724087 0.87 LMNA (0.75) LMNASIGMAR1POLBMAPK1CYP1A2
SCHEMBL13479679 0.85 LMNA (0.74) LMNASIGMAR1POLBMAPK1L3MBTL1
SCHEMBL8587899 0.83 LMNA (0.71) LMNASIGMAR1POLBMAPK1CYP1A2
SCHEMBL13995787 0.83 LMNA (0.71) LMNASIGMAR1POLBMAPK1CYP3A4
SCHEMBL18313993 0.81 LMNA (0.69) LMNASIGMAR1POLBMAPK1CYP1A2
SCHEMBL19772457 0.81 LMNA (0.68) LMNAPOLBMAPK1CYP3A4CYP2D6
SCHEMBL11261490 0.80 LMNA (0.67) LMNASIGMAR1POLBMAPK1CYP1A2
SCHEMBL11261494 0.80 LMNA (0.67) LMNASIGMAR1POLBMAPK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3167 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
US-20250122274-A1 SELECTIVE AND POTENT INHIBITORY ANTIBODIES OF MYOSTATIN ACTIVATION SCHOLAR ROCK, INC. 2025-04-17 US claimed
WO-2025042770-A1 ANOREXIA-SENSITIZING AGENTS THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2025-02-27 WO claimed
CN-119233997-A Tetrahedral antibodies 生物分子控股有限责任公司 2024-12-31 CN claimed
EP-4463485-A2 TETRAHEDRAL ANTIBODIES Biomolecular Holdings LLC (US) 2024-11-20 EP claimed
CN-118384290-A Hybrid immunoglobulins containing non-peptide linkages 生物分子控股有限责任公司 2024-07-26 CN claimed
US-20240075043-A1 IMMEDIATE AND CONTROLLED RELEASE APPETITE SUPPRESSANT COMPOSITIONS FOR WEIGHT LOSS Red Mountain Med Spa, LLC (US) 2024-03-07 US claimed
WO-2023137373-A1 TETRAHEDRAL ANTIBODIES BIOMOLECULAR HOLDINGS LLC (US) 2023-07-20 WO claimed
WO-2023137387-A2 TETRAHEDRAL ANTIBODIES BIOMOLECULAR HOLDINGS LLC (US) 2023-07-20 WO claimed
US-20230220115-A1 TETRAHEDRAL ANTIBODIES BIOMOLECULAR HOLDINGS LLC (US) 2023-07-13 US claimed
US-20030114495-A1 Substituted imidazoles as cannabinoid receptor modulators MERCK SHARP & DOHME CORP. 2003-06-19 US claimed
WO-2003045313-A2 2-AMINOQUINOLINE COMPOUNDS MERCK & CO. INC. (US) 2003-06-05 WO claimed
WO-2003045920-A1 4-AMINOQUINOLINE COMPOUNDS MERCK & CO., INC. (US) 2003-06-05 WO claimed
WO-2003007887-A2 SUBSTITUTED IMIDAZOLES AS CANNABINOID RECEPTOR MODULATORS MERCK & CO., INC. (US) 2003-01-30 WO claimed
JP-2001524960-A 2001-12-04 JP claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
EP-0977572-A1 USE OF NK-1 RECEPTOR ANTAGONISTS FOR TREATING EATING DISORDERS MERCK SHARP & DOHME LTD. (GB) 2000-02-09 EP claimed
WO-1998047513-A1 USE OF NK-1 RECEPTOR ANTAGONISTS FOR TREATING EATING DISORDERS MERCK SHARP & DOHME LIMITED (GB) 1998-10-29 WO claimed