Miroprofen

Miroprofen

SCHEMBL26767

CC(C(=O)O)c1ccc(-c2cn3ccccc3n2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 1.00
PTGS1 P23219 1/20 1.00
RAB9A P51151 11/20 0.58
NPC1 O15118 11/20 0.58
KDM4E B2RXH2 10/20 0.58
GFER P55789 3/20 0.58
HDAC6 Q9UBN7 1/20 0.56
POLB P06746 2/20 0.56
PKM P14618 4/20 0.56
EPHX2 P34913 1/20 0.56
ALDH1A1 P00352 7/20 0.53
SMN1; SMN2 Q16637 7/20 0.53
HPGD P15428 3/20 0.53
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
GAA P10253 1/20 0.52
MIF P14174 1/20 0.52
MAPK1 P28482 2/20 0.52
MAPT P10636 3/20 0.51
NPSR1 Q6W5P4 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Miroprofen SCHEMBL11832509 0.99 PTGS2 (0.97) PTGS2PTGS1RAB9ANPC1KDM4E
SCHEMBL12608963 0.92 PTGS1 (0.85) PTGS2PTGS1RAB9ANPC1KDM4E
SCHEMBL11819076 0.88 PTGS1 (0.79) PTGS2PTGS1RAB9ANPC1KDM4E
SCHEMBL11822617 0.88 PTGS1 (0.79) PTGS2PTGS1RAB9ANPC1KDM4E
Miroprofen SCHEMBL3059150 0.87 PTGS2 (0.76) PTGS2PTGS1RAB9ANPC1KDM4E
SCHEMBL11822336 0.84 PTGS1 (0.72) PTGS2PTGS1RAB9ANPC1KDM4E
SCHEMBL2431742 0.83 PTGS1 (0.71) PTGS2PTGS1RAB9ANPC1KDM4E
SCHEMBL2739322 0.83 PTGS1 (0.71) PTGS2PTGS1RAB9ANPC1KDM4E
SCHEMBL15486399 0.81 PTGS1 (0.68) PTGS2PTGS1RAB9ANPC1KDM4E
SCHEMBL11818001 0.81 PTGS1 (0.67) PTGS2PTGS1RAB9ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8834 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260000741-A1 METHOD OF AMELIORATING A PRO-INFLAMMATORY IMMUNOPHENOTYPE IN FARBER DISEASE SUBJECTS BY REPEATED ADMINISTRATION OF A RECOMBINANT HUMAN ACID CERAMIDASE ACERAGEN INC (US) 2026-01-01 US claimed
EP-4470565-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT OnQuality Pharmaceuticals China Ltd. (CN) 2024-12-04 EP claimed
US-RE50218-E1 Non-steroidal anti-inflammatory ophthalmic compositions SUN PHARMACEUTICAL INDUSTRIES LIMITED (IN) 2024-11-26 US claimed
CN-118742325-A Methods for preventing or treating diseases or conditions associated with antineoplastic agents 上海岸阔医药科技有限公司 2024-10-01 CN claimed
EP-4308063-A1 PRE-FILLING SYSTEM TO ELIMINATE BUBBLES INSIDE CAPSULES HAVING A SOLID DOSAGE FORM Procaps SA (US) 2024-01-24 EP claimed
EP-3752201-B1 SUSPENSION OF NANOSCALE, ORGANIC PARTICLES AND PROCESS FOR PRODUCTION THEREOF UNIV FRIEDRICH ALEXANDER ER (DE) 2023-11-22 EP claimed
WO-2023142996-A1 METHOD FOR PREVENTING OR TREATING DISEASE OR DISORDER ASSOCIATED WITH ANTINEOPLASTIC AGENT 上海岸阔医药科技有限公司 2023-08-03 WO claimed
EP-4185277-A1 SOFT SHELL GELATIN CAPSULES Procaps SA (US) 2023-05-31 EP claimed
US-20230088240-A1 ACCELERATING THE DRYING RATE OF SOFTGEL CAPSULES GLAS AMERICAS LLC 2023-03-23 US claimed
WO-2022197983-A1 PRE-FILLING SYSTEM TO ELIMINATE BUBBLES INSIDE CAPSULES HAVING A SOLID DOSAGE FORM PROCAPS SA (US) 2022-09-22 WO claimed
EP-0167566-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING XANTHINES AND METHODS OF USING SAME SUNSHINE, Abraham (US) 1986-01-15 EP claimed
US-4552899-A ANTITUSSIVE AGENTS ANALGESIC ASSOCIATES (US) 1985-11-12 US claimed
WO-1985004589-A1 COUGH/COLD MIXTURES COMPRISING NON-STEROIDAL ANTI-INFLAMMATORY DRUGS SUNSHINE ABRAHAM 1985-10-24 WO claimed
WO-1985003443-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING DIPHENHYDRAMINE AND METHODS OF USING SAME RICHARDSON-VICKS, INC. (US) 1985-08-15 WO claimed
WO-1985002542-A1 ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING XANTHINES AND METHODS OF USING SAME SUNSHINE ABRAHAM 1985-06-20 WO claimed
US-4522826-A SYNERGISTIC MIXTURES RICHARDSON-VICKS INC. (US) 1985-06-11 US claimed
US-4486436-A Analgesic and anti-inflammatory compositions comprising caffeine and methods of using same ANALGESIC ASSOCIATES (US) 1984-12-04 US claimed
EP-0114886-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE. SUNSHINE ABRAHAM (US) 1984-08-08 EP claimed
WO-1984000490-A1 IMPROVED ANALGESIC AND ANTI-INFLAMMATORY COMPOSITIONS COMPRISING CAFFEINE AND METHODS OF USING SAME SUNSHINE ABRAHAM 1984-02-16 WO claimed
US-3978071-A ANALGESIC, ANTIPYRETIC, ANTIINFLAMMATORY YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JA) 1976-08-31 US claimed