SCHEMBL2679366

SCHEMBL2679366

CNc1nccc(-c2cc(NCC(=O)Nc3nc4ccccc4n3C)c3cc(OC)ccc3c2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.42
PLK1 P53350 2/20 0.42
PTK2 Q05397 2/20 0.42
AURKB Q96GD4 2/20 0.42
AKT1 P31749 1/20 0.42
NPC1 O15118 4/20 0.41
RAB9A P51151 4/20 0.41
TEK Q02763 1/20 0.41
PKM P14618 1/20 0.40
NR1I2 O75469 1/20 0.38
TP53 P04637 1/20 0.37
MKNK2 Q9HBH9 4/20 0.37
MKNK1 Q9BUB5 3/20 0.37
MGLL Q99685 1/20 0.37
NTRK1 P04629 2/20 0.36
NTRK2 Q16620 2/20 0.36
HDAC3 O15379 1/20 0.36
NCOR1 O75376 1/20 0.36
HDAC2 Q92769 1/20 0.36
TSHR P16473 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6128762 0.94 NPC1 (0.43) KDRPLK1PTK2AURKBAKT1
SCHEMBL2679375 0.86 HDAC3 (0.41) KDRAURKBAKT1TEKMKNK1
SCHEMBL6128802 0.83 HDAC3 (0.43) KDRAURKBTEKTP53MKNK1
SCHEMBL2678820 0.82 MEN1 (0.42) MKNK1MGLLHDAC3NCOR1HDAC2
SCHEMBL2678140 0.81 HDAC3 (0.46) PKMHDAC3NCOR1HDAC2MEN1
SCHEMBL2679120 0.80 HDAC3 (0.38) AKT1HDAC3NCOR1HDAC2HTT
SCHEMBL2678111 0.80 MTNR1A (0.40) HDAC3NCOR1HDAC2
SCHEMBL2678527 0.79 MTNR1A (0.39) KDRTEKHDAC3NCOR1HDAC2
SCHEMBL6128580 0.79 HDAC3 (0.40) MKNK1MGLLHDAC3NCOR1HDAC2
SCHEMBL2175597 0.78 HDAC3 (0.39) AKT1HDAC3NCOR1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8173808-B2 Substituted naphthalenyl-pyrimidine compounds ARQULE, INC. (US) 2012-05-08 US claimed