SCHEMBL2679375

SCHEMBL2679375

CNc1nccc(-c2cc(NCC(=O)Nc3ncccn3)c3cc(OC)ccc3c2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.41
NCOR1 O75376 1/20 0.41
HDAC2 Q92769 1/20 0.41
PIK3CA P42336 4/20 0.39
PIK3CG P48736 3/20 0.39
PIK3CB P42338 2/20 0.39
DYRK1A Q13627 4/20 0.39
CLK4 Q9HAZ1 4/20 0.39
DYRK1B Q9Y463 3/20 0.39
ABL1 P00519 1/20 0.38
BCR P11274 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RIOK2 Q9BVS4 2/20 0.38
GSK3A P49840 1/20 0.38
MAPK10 P53779 1/20 0.38
CLK1 P49759 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6128802 0.93 HDAC3 (0.43) HDAC3NCOR1HDAC2PIK3CAPIK3CG
SCHEMBL2678820 0.90 MEN1 (0.42) HDAC3NCOR1HDAC2PIK3CAPIK3CG
SCHEMBL2678140 0.89 HDAC3 (0.46) HDAC3NCOR1HDAC2PIK3CAPIK3CG
SCHEMBL2679120 0.88 HDAC3 (0.38) HDAC3NCOR1HDAC2PIK3CAPIK3CG
SCHEMBL2678111 0.87 MTNR1A (0.40) HDAC3NCOR1HDAC2PIK3CAPIK3CG
SCHEMBL2678527 0.86 MTNR1A (0.39) HDAC3NCOR1HDAC2PIK3CAPIK3CG
SCHEMBL6128580 0.86 HDAC3 (0.40) HDAC3NCOR1HDAC2PIK3CAPIK3CG
SCHEMBL2679366 0.86 KDR (0.42) HDAC3NCOR1HDAC2SMN1; SMN2AKT1
SCHEMBL6128566 0.85 HDAC3 (0.46) HDAC3NCOR1HDAC2PIK3CAPIK3CG
SCHEMBL2178808 0.85 CASP2 (0.41) HDAC3NCOR1HDAC2PIK3CAPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8173808-B2 Substituted naphthalenyl-pyrimidine compounds ARQULE, INC. (US) 2012-05-08 US claimed