SCHEMBL26812005

SCHEMBL26812005

CCOc1ccc(S(=O)(=O)Nc2ccc(C(=O)N3CCN(c4ccccc4OC)CC3)cc2)cc1OCC

nearest known ligand 0.75

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 1/20 0.75
PKM P14618 4/20 0.75
ALDH1A1 P00352 4/20 0.73
MAPT P10636 2/20 0.73
HTT P42858 2/20 0.73
TSHR P16473 2/20 0.57
LMNA P02545 2/20 0.56
GAA P10253 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
KDM4E B2RXH2 1/20 0.56
RECQL P46063 1/20 0.56
REV1 Q9UBZ9 1/20 0.55
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
USP2 O75604 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
HSD17B10 Q99714 1/20 0.54
POLB P06746 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19036159 0.86 PKM (0.83) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL2704273 0.85 PKM (0.78) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL2702167 0.85 PKM (0.82) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL12964838 0.85 PKM (1.00) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL2703016 0.85 ALDH1A1 (0.86) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL12976972 0.85 ALDH1A1 (0.86) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL10008458 0.85 HCRTR1 (0.73) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL2702638 0.83 PKM (0.84) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL2703621 0.83 ALDH1A1 (0.74) HCRTR1PKMALDH1A1MAPTHTT
SCHEMBL12235 0.82 PKM (0.60) HCRTR1PKMALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3406251-B1 PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY AGIOS PHARMACEUTICALS INC (US) 2023-11-29 EP disclosed