SCHEMBL2683560

SCHEMBL2683560

FC(F)(F)c1ccc(/C(=C/c2ccc(Br)cc2)c2ccc(Br)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 4/20 0.50
PTGS2 P35354 2/20 0.50
NQO2 P16083 1/20 0.50
ESR1 P03372 1/20 0.47
ESR2 Q92731 1/20 0.47
GPR183 P32249 1/20 0.47
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
HPGD P15428 1/20 0.42
AKR1C3 P42330 1/20 0.41
HDAC3 O15379 1/20 0.41
ADAM17 P78536 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2683562 1.00 PTGS1 (0.50) PTGS1PTGS2NQO2ESR1ESR2
SCHEMBL28816901 0.89 KIF11 (0.47) PTGS1PTGS2NQO2ESR1ESR2
SCHEMBL28816900 0.89 KIF11 (0.47) PTGS1PTGS2NQO2ESR1ESR2
SCHEMBL9937304 0.87 PTGS1 (0.43) PTGS1PTGS2NQO2ESR1ESR2
SCHEMBL21738730 0.84 ESR1 (0.62) PTGS2ESR1ESR2CES2CES1
SCHEMBL2683558 0.82 ESR1 (0.47) PTGS2ESR1ESR2GPR183KDM4E
SCHEMBL2683557 0.82 ESR1 (0.47) PTGS2ESR1ESR2GPR183KDM4E
SCHEMBL9937306 0.82 PTGS1 (0.39) PTGS1PTGS2NQO2ESR1ESR2
SCHEMBL1746513 0.77 GSK3B (0.43) GPR183CES2CES1HDAC1HDAC8
SCHEMBL1746517 0.77 GSK3B (0.43) GPR183CES2CES1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140155382-A1 ANTI-VIRAL COMPOUNDS ABBVIE INC. (US) 2014-06-05 US disclosed
US-20120115918-A1 Anti-Viral Compounds ABBOTT LABORATORIES (US) 2012-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120115918-A1 Anti-Viral Compounds HAVCR2, EIF2AK2, MAVS PTGS1 1687/4885PTGS2 2159/4885NQO2 2381/4885
US-20140155382-A1 ANTI-VIRAL COMPOUNDS HAVCR2, EIF2AK2, MAVS PTGS1 1687/4885PTGS2 2159/4885NQO2 2381/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.