SCHEMBL2693397

SCHEMBL2693397

CCCN(CCC)[C@H]1CCCN(Cc2ccc(S(=O)(=O)N(Cc3ncc[nH]3)Cc3ncc[nH]3)cc2)C1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
CXCR4 P61073 3/20 0.37
KAT2B Q92831 1/20 0.37
BCHE P06276 1/20 0.37
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HTT P42858 1/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HTR2B P41595 1/20 0.34
EP300 Q09472 1/20 0.34
HIF1A Q16665 1/20 0.34
ROCK2 O75116 2/20 0.34
CTSD P07339 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2694615 0.82 CXCR4 (0.54) ALDH1A1CXCR4KAT2BBCHEHTT
SCHEMBL2693687 0.77 CXCR4 (0.37) CXCR4HTT
SCHEMBL4778325 0.77 TAS2R14 (0.38) ALDH1A1CXCR4LMNA
SCHEMBL4778306 0.77 TAS2R14 (0.38) ALDH1A1CXCR4LMNA
SCHEMBL2693691 0.77 CXCR4 (0.37) CXCR4HTT
Hydrochloric Acid SCHEMBL2695183 0.76 TAS2R14 (0.38) ALDH1A1CXCR4LMNA
Hydrochloric Acid SCHEMBL2695170 0.76 TAS2R14 (0.38) ALDH1A1CXCR4LMNA
SCHEMBL2695476 0.73 CXCR4 (0.35) ALDH1A1CXCR4LMNA
SCHEMBL2695473 0.73 CXCR4 (0.35) ALDH1A1CXCR4LMNA
SCHEMBL2695586 0.72 CA12 (0.33) CXCR4KAT2BMEN1KMT2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8519124-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2013-08-27 US disclosed
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2012-08-16 US disclosed
US-8168783-B2 Chemokine receptor antagonists and use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2012-05-01 US disclosed
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD., (JP) 2009-07-02 US disclosed
EP-1961744-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2008-08-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090169567-A1 BASIC GROUP-CONTAINING COMPOUND AND USE THEREOF CXCR4, CXCL12, CXCR3 ALDH1A1 470/4885CXCR4 1/4885KAT2B 3346/4885
US-20120207765-A1 CHEMOKINE RECEPTOR ANTAGONISTS AND USE THEREOF CXCR4, CXCR3, CXCR1 ALDH1A1 893/4885CXCR4 1/4885KAT2B 3493/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.