SCHEMBL26995231

SCHEMBL26995231

CCOC(=O)C(Cc1cccc(OC(F)(F)F)c1)N=C(c1ccccc1)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 1/20 0.45
MAPK14 Q16539 1/20 0.44
AAK1 Q2M2I8 1/20 0.44
ELANE P08246 1/20 0.42
PPARG P37231 5/20 0.41
PPARA Q07869 4/20 0.41
GPR139 Q6DWJ6 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PTGER4 P35408 1/20 0.40
PTGER2 P43116 1/20 0.40
EPHX2 P34913 1/20 0.40
CYP2C9 P11712 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
CYP4X1 Q8N118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31506282 1.00 TRPM8 (0.45) TRPM8MAPK14AAK1ELANEPPARG
SCHEMBL395095 0.89 MRGPRX4 (0.42) AAK1PPARGPPARAMRGPRX4TSHR
SCHEMBL30831623 0.88 TRPM8 (0.49) TRPM8MAPK14AAK1PPARGPPARA
SCHEMBL30831587 0.88 TAAR1 (0.45) MRGPRX4TSHRMAPK1TDP1L3MBTL1
SCHEMBL23436 0.88 TAAR1 (0.45) MRGPRX4TSHRMAPK1TDP1L3MBTL1
SCHEMBL18833 0.88 TAAR1 (0.45) MRGPRX4TSHRMAPK1TDP1L3MBTL1
SCHEMBL18482288 0.80 AAK1 (0.45) AAK1PPARGPPARAMRGPRX4EPHX2
SCHEMBL26995244 0.79 RAB9A (0.47) MRGPRX4MAPK1L3MBTL1
SCHEMBL30831549 0.79 RAB9A (0.47) MRGPRX4MAPK1L3MBTL1
SCHEMBL5311248 0.78 AAK1 (0.42) AAK1PPARGEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024008941-A1 NEW SPIROCYCLOHEXANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS ANTI-APOPTOTIC INHIBITORS LES LABORATOIRES SERVIER (FR) 2024-01-11 WO disclosed