SCHEMBL27002575

SCHEMBL27002575

CCOC(=O)c1ccc2nc(-c3ccncc3)[nH]c2c1.CCOC(=O)c1ccc2nc(-c3ccncc3)[nH]c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 2/20 1.00
PKN2 Q16513 2/20 1.00
SIRT2 Q8IXJ6 6/20 0.77
SIRT1 Q96EB6 5/20 0.77
SIRT3 Q9NTG7 2/20 0.77
ATM Q13315 1/20 0.58
ALOX5 P09917 1/20 0.58
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58
IMPDH2 P12268 1/20 0.58
CHEK2 O96017 5/20 0.57
KDM4E B2RXH2 1/20 0.55
ALDH1A1 P00352 1/20 0.55
GAA P10253 1/20 0.55
HPGD P15428 1/20 0.55
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19994427 1.00 PKN1 (1.00) PKN1PKN2SIRT2SIRT1SIRT3
SCHEMBL19994531 0.87 SIRT2 (0.79) PKN1PKN2SIRT2SIRT1SIRT3
SCHEMBL19994496 0.83 SIRT2 (0.72) PKN1PKN2SIRT2SIRT1SIRT3
SCHEMBL2807193 0.83 CHEK2 (0.73) PKN1PKN2SIRT2SIRT1SIRT3
SCHEMBL6169071 0.80 PKN1 (0.67) PKN1PKN2SIRT2SIRT1SIRT3
SCHEMBL4259320 0.80 PKN1 (0.77) PKN1PKN2NPC1RAB9ACHEK2
SCHEMBL2357098 0.80 CHEK2 (0.74) PKN1PKN2SIRT2SIRT1SIRT3
SCHEMBL8248442 0.79 PKN1 (0.65) PKN1PKN2SIRT2SIRT1SIRT3
SCHEMBL17275543 0.79 PKN1 (0.65) PKN1PKN2SIRT2SIRT1SIRT3
SCHEMBL9261347 0.79 ALDH1A1 (0.74) PKN1PKN2SIRT2SIRT1SIRT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3515904-B1 BENZOIMIDAZOLE DERIVATIVES AS ANTICANCER AGENTS CENTRE LEON BERARD (FR) 2024-01-17 EP disclosed