SCHEMBL270119

SCHEMBL270119

O=C(C=CCCC=CC(=O)NO)NO

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 10/20 0.39
HDAC2 Q92769 9/20 0.39
HDAC3 O15379 9/20 0.39
HDAC8 Q9BY41 9/20 0.39
HDAC1 Q13547 9/20 0.39
HDAC4 P56524 5/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
CNR1 P21554 2/20 0.36
CNR2 P34972 2/20 0.36
TRPA1 O75762 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
HDAC10 Q969S8 5/20 0.35
HDAC11 Q96DB2 5/20 0.35
HDAC5 Q9UQL6 5/20 0.35
HDAC7 Q8WUI4 4/20 0.35
HDAC9 Q9UKV0 4/20 0.35
ADAM17 P78536 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9716525 0.87
SCHEMBL8089117 0.85
SCHEMBL8089108 0.81 PSMB11 (0.45) TAS1R3TAS1R1CNR1CNR2
SCHEMBL5791476 0.79 PSMB11 (0.51) CNR1CNR2
SCHEMBL5791472 0.79 PSMB11 (0.51) CNR1CNR2
SCHEMBL13971007 0.78 HDAC2 (0.67) HDAC6HDAC2HDAC3HDAC8HDAC1
SCHEMBL2356012 0.78
SCHEMBL5794871 0.78 PSMB11 (0.54) CNR1CNR2
SCHEMBL5794870 0.78 PSMB11 (0.54) CNR1CNR2
SCHEMBL8089119 0.78 PSMB11 (0.54) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 156 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728339-B1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS AMO Ireland (IE) 2022-07-06 EP claimed
US-11359031-B2 Composition for ophthalmological products Johnson & Johnson Surgical Vision, Inc. (US) 2022-06-14 US claimed
EP-3200840-B1 LOW-WATER CONTENT ACRYLATE-ACRYLAMIDE COPOLYMERS FOR OPHTHALMIC DEVICES ALCON INC (CH) 2021-11-17 EP claimed
EP-3728339-A1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS Merck Patent GmbH (DE) 2020-10-28 EP claimed
US-20200332041-A1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS MERCK PATENT GMBH (DE) 2020-10-22 US claimed
EP-3200839-B1 HYDROPHOBIC ACRYLATE-ACRYLAMIDE COPOLYMERS FOR OPHTHALMIC DEVICES NOVARTIS AG (CH) 2019-09-04 EP claimed
EP-3502147-A1 COMPOSITION FOR OPHTHALMOLOGICAL PRODUCTS Merck Patent GmbH (DE) 2019-06-26 EP claimed
EP-3223870-B1 WET-PACK INTRAOCULAR LENS MATERIALS WITH HIGH REFRACTIVE INDEX NOVARTIS AG (CH) 2018-09-26 EP claimed
EP-1444239-B1 HIGH REFRACTIVE INDEX AROMATIC-BASED SILYL MONOMERS BAUSCH & LOMB (US) 2008-12-24 EP claimed
EP-1448571-B1 HIGH REFRACTIVE INDEX AROMATIC-BASED SILOXANE MONOFUNCTIONAL MACROMONOMERS BAUSCH & LOMB (US) 2008-05-21 EP claimed
EP-0425436-B1 Reactive silicone and/or fluorine containing hydrophilic prepolymers and polymers thereof CIBA GEIGY AG (CH) 1996-12-27 EP claimed
EP-0421264-B1 Hydrophilic swellable polymers CASSELLA FARBWERKE MAINKUR AG (DE) 1994-08-10 EP claimed
US-5236965-A Absorbers, acrylic CASSELLA AKTIENGESELLSCHAFT (DE) 1993-08-17 US claimed
US-5214075-A Used as absorption agents for water and aqueous solutions CASSELLA AKTIENGESELLSCHAFT (DE) 1993-05-25 US claimed
US-5182312-A Crosslinked acrylic polymer foams CASSELLA AKTIENGESELLSCHAFT (DE) 1993-01-26 US claimed
US-4539200-A CLEANING WOUNDS CROSSLINKED POLYAMIDES THE KENDALL COMPANY (US) 1985-09-03 US claimed
WO-2025022004-A2 OPHTHALMIC LENS CONTAMAC LIMITED (GB) 2025-01-30 WO disclosed
EP-4182737-B1 OPTICALLY ACTIVE DEVICES AMO Ireland (IE) 2024-07-03 EP disclosed
US-3992324-A GROUP 8 AND 6B OXIDES OR SULFIDES LABOFINA S.A. (BE) 1976-11-16 US disclosed
US-3966996-A ADDITION POLYMERIZATION, DISPERSION LABOFINA S.A. (BE) 1976-06-29 US disclosed