SCHEMBL27100910

SCHEMBL27100910

Cc1c(Br)c(Cl)cc2c(N3CCCCCC3)nc(Cl)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 2/20 0.38
LMNA P02545 1/20 0.38
PRNP P04156 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
PPARG P37231 1/20 0.38
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
NR2E3 Q9Y5X4 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
CHRM4 P08173 2/20 0.38
PDE10A Q9Y233 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TP53 P04637 2/20 0.36
MAT2A P31153 1/20 0.35
GLP1R P43220 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17030874 0.84 SMN1; SMN2 (0.44) SMN1; SMN2ALDH1A1MAPTLMNAPRNP
SCHEMBL27147161 0.84 SMN1; SMN2 (0.44) SMN1; SMN2ALDH1A1MAPTLMNAPRNP
SCHEMBL30922651 0.76 SMN1; SMN2 (0.44) SMN1; SMN2ALDH1A1MAPTLMNAPRNP
SCHEMBL38660623 0.75 GPR35 (0.33)
SCHEMBL19422066 0.74 SMN1; SMN2 (0.47) SMN1; SMN2HTTKMT2A
SCHEMBL25720390 0.74 SMN1; SMN2 (0.47) SMN1; SMN2HTTKMT2A
SCHEMBL25081570 0.73 SMN1; SMN2 (0.43) SMN1; SMN2ALDH1A1MAPTLMNATSHR
SCHEMBL31470355 0.72 ALDH1A1 (0.34) SMN1; SMN2ALDH1A1MAT2A
SCHEMBL19695842 0.71 HTR2C (0.40) MAPTHTTMEN1KMT2A
SCHEMBL25253238 0.71 ALDH1A1 (0.33) SMN1; SMN2ALDH1A1TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024044667-A2 SMALL MOLECULE INHIBITORS OF KRAS PROTEINS MERCK SHARP & DOHME LLC (US) 2024-02-29 WO disclosed