SCHEMBL2710461

SCHEMBL2710461

BrCCCC(Br)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.40
HRH1 P35367 6/20 0.40
SIGMAR1 Q99720 1/20 0.38
TRPA1 O75762 2/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
TAAR1 Q96RJ0 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
DPP4 P27487 2/20 0.33
MTOR P42345 1/20 0.33
RAB9A P51151 1/20 0.33
GRM7 Q14831 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
F2 P00734 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22042217 0.88 HRH1 (0.44) HTR2AHRH1SIGMAR1TRPA1CES2
SCHEMBL4450297 0.86 HRH1 (0.41) HTR2AHRH1SIGMAR1TRPA1CES2
SCHEMBL22042211 0.83 HRH1 (0.46) HTR2AHRH1TRPA1CES2CES1
SCHEMBL14307122 0.82 HTR2A (0.40) HTR2AHRH1SIGMAR1TRPA1CES2
SCHEMBL904449 0.81 HRH1 (0.60) HTR2AHRH1SIGMAR1TAAR1
SCHEMBL3841684 0.80 HTR2A (0.36) HTR2A
SCHEMBL9789913 0.80 HTR2A (0.65) HTR2AHRH1TAAR1TSHR
SCHEMBL4889343 0.80 HTR2A (0.39) HTR2AHRH1SIGMAR1TRPA1CES2
SCHEMBL1920593 0.80 POLB (0.45) HTR2AHRH1SIGMAR1ALDH1A1
SCHEMBL1308306 0.78 TRPA1 (0.40) HTR2AHRH1SIGMAR1TRPA1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed
US-3992251-A Process of making wet strength paper containing mono primary polyamine and organic dihalide modified, epoxidized polyamide DIAMOND SHAMROCK CORPORATION (US) 1976-11-16 US disclosed