SCHEMBL2712232

SCHEMBL2712232

COC(=O)c1cc(C(=O)OC(C)(C)C)cc(N2CCCC2=O)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
ALDH1A1 P00352 5/20 0.37
HPGD P15428 3/20 0.37
GAA P10253 2/20 0.37
KDM4E B2RXH2 2/20 0.37
GLA P06280 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
SRD5A1 P18405 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MAPT P10636 1/20 0.35
TYK2 P29597 2/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2712897 0.97 ADORA2A (0.36) ADORA2AADORA1ALDH1A1HPGDGAA
SCHEMBL2711845 0.88 ALDH1A1 (0.43) ADORA2AADORA1ALDH1A1HPGDGAA
SCHEMBL2712767 0.86 ALDH1A1 (0.42) ADORA2AADORA1ALDH1A1HPGDKDM4E
SCHEMBL5853270 0.85 ALDH1A1 (0.41) ADORA2AADORA1ALDH1A1HPGDGAA
SCHEMBL2712965 0.83 KDM4E (0.40) ALDH1A1GAAKDM4EMEN1KMT2A
SCHEMBL6465278 0.82 MAP4K1 (0.37) SRD5A1TYK2USP30
SCHEMBL5221158 0.79 MEN1 (0.48) ALDH1A1HPGDGAAKDM4EMEN1
SCHEMBL2712865 0.79 HDAC1 (0.34) ALDH1A1GLAUCHL1USP30
SCHEMBL22425776 0.77 ADORA2A (0.42) ADORA2AADORA1ALDH1A1HPGDGAA
SCHEMBL2711600 0.75 HPGD (0.38) ADORA1ALDH1A1HPGDGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed