SCHEMBL27133166

SCHEMBL27133166

NC(CCN(Cc1ccc(-c2cccs2)s1)Cc1ccc(-c2cccs2)s1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.47
DPP4 P27487 3/20 0.46
SLC1A5 Q15758 12/20 0.42
ALOX5 P09917 1/20 0.40
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
LMNA P02545 1/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26987838 1.00 LTA4H (0.47) LTA4HDPP4SLC1A5ALOX5KDM4E
SCHEMBL26987958 0.84 HDAC3 (0.55) SLC1A5HDAC3HDAC1HDAC2HDAC8
SCHEMBL27125342 0.84 HDAC3 (0.55) SLC1A5HDAC3HDAC1HDAC2HDAC8
SCHEMBL27125658 0.83 CYP2C19 (0.49) SLC1A5ALDH1A1
SCHEMBL26987705 0.83 CYP2C19 (0.49) SLC1A5ALDH1A1
SCHEMBL27131855 0.79 SLC1A5 (0.74) SLC1A5
SCHEMBL26987832 0.79 SLC1A5 (0.74) SLC1A5
SCHEMBL26987594 0.70 NNMT (0.54) SLC1A5
SCHEMBL27130058 0.70 NNMT (0.54) SLC1A5
SCHEMBL9584558 0.70 CYP2C19 (0.56) ALDH1A1NPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024010732-A1 SMALL MOLECULE INHIBITORS OF GLUTAMINE TRANSPORTER ASCT2 AND METHODS OF USE THEREOF BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2024-01-11 WO disclosed