SCHEMBL2714979

SCHEMBL2714979

NC(=O)c1cc(F)cnc1Nc1cccc(-c2ncccn2)c1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.59
SYK P43405 13/20 0.54
NPC1 O15118 2/20 0.46
MAPT P10636 2/20 0.46
RAB9A P51151 2/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
KMT2A Q03164 1/20 0.46
KCNH2 Q12809 1/20 0.46
FGFR3 P22607 1/20 0.43
KDR P35968 1/20 0.43
SIRT2 Q8IXJ6 1/20 0.42
SIRT1 Q96EB6 1/20 0.42
JAK2 O60674 1/20 0.42
AHR P35869 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CSF1R P07333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2714471 0.84 LMNA (0.70) LMNASYKNPC1MAPTRAB9A
SCHEMBL8179361 0.80 LMNA (0.47) LMNASYKFGFR3KDRSIRT2
SCHEMBL16202719 0.78 SYK (0.67) SYKKCNH2
SCHEMBL870223 0.78 DHODH (0.53) LMNAMEN1ALDH1A1KMT2ASIRT2
SCHEMBL2627254 0.75 SYK (0.63) SYKKCNH2
SCHEMBL9496511 0.75 LMNA (1.00) LMNASYKNPC1MAPTRAB9A
SCHEMBL2715102 0.74 SYK (0.57) SYK
SCHEMBL2714322 0.74 SYK (0.57) SYK
SCHEMBL2716760 0.73 SYK (0.63) LMNASYKKCNH2
SCHEMBL2716764 0.73 SYK (0.63) LMNASYKKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2635556-A2 BENZAMIDES AND NICOTINAMIDES AS SYK MODULATORS Portola Pharmaceuticals, Inc. (US) 2013-09-11 EP claimed
WO-2012061418-A2 BENZAMIDES AND NICOTINAMIDES AS SYK MODULATORS PORTOLA PHARMACEUTICALS, INC. (US) 2012-05-10 WO claimed