SCHEMBL27165232

SCHEMBL27165232

CCOCCOc1ccc(C[C@H]2CN(CC(=O)[O-])CCN(CC(=O)[O-])CCN(CC(=O)O)CCN2CC(=O)[O-])cc1.[Gd+3]

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
FOLH1 Q04609 1/20 0.37
HRH1 P35367 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 3/20 0.36
TDP1 Q9NUW8 1/20 0.36
S1PR1 P21453 3/20 0.35
S1PR5 Q9H228 3/20 0.35
ADORA3 P0DMS8 1/20 0.35
HTR2A P28223 1/20 0.35
HTR7 P34969 1/20 0.35
OPRM1 P35372 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
MMP3 P08254 1/20 0.35
MMP9 P14780 1/20 0.35
ADAM17 P78536 1/20 0.35
S1PR3 Q99500 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27166218 0.99 KDM4E (0.38) MEN1KMT2AFOLH1HRH1KDM4E
SCHEMBL27166222 0.99 KDM4E (0.38) MEN1KMT2AFOLH1HRH1KDM4E
SCHEMBL27166229 0.92 KDM4E (0.40) MEN1KMT2AFOLH1HRH1KDM4E
SCHEMBL27166228 0.92 FOLH1 (0.36) MEN1KMT2AFOLH1KDM4EALDH1A1
SCHEMBL27166220 0.92 FOLH1 (0.36) MEN1KMT2AFOLH1KDM4EALDH1A1
SCHEMBL27166219 0.92 MEN1 (0.46) MEN1KMT2AFOLH1KDM4EALDH1A1
SCHEMBL27166254 0.91 KDM4E (0.41) MEN1KMT2AFOLH1HRH1KDM4E
SCHEMBL27165218 0.91 ALDH1A1 (0.43) MEN1KMT2AFOLH1KDM4EALDH1A1
SCHEMBL27166241 0.91 KDM4E (0.41) MEN1KMT2AFOLH1HRH1KDM4E
SCHEMBL27166221 0.91 ALDH1A1 (0.43) MEN1KMT2AFOLH1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4567716-B1 GENERATING SYNTHETIC REPRESENTATIONS BAYER AG (DE) 2026-05-13 EP claimed
EP-4567715-B1 GENERATING SYNTHETIC REPRESENTATIONS BAYER AG (DE) 2026-05-13 EP claimed
EP-4581641-B1 GENERATION OF SYNTHETIC RADIOLOGICAL RECORDINGS BAYER AG (DE) 2026-05-06 EP claimed
EP-4581640-B1 GENERATION OF SYNTHETIC RADIOLOGICAL RECORDINGS BAYER AG (DE) 2026-04-22 EP claimed
EP-4485474-B1 GENERATION OF ARTIFICIAL CONTRAST ENHANCED RADIOLOGICAL RECORDINGS BAYER AG (DE) 2026-04-08 EP claimed
US-20260051027-A1 GENERATION OF SYNTHETIC CONTRAST-ENHANCED RADIOLOGICAL IMAGES BAYER AG (DE) 2026-02-19 US claimed
EP-4664393-A1 GENERATION OF SYNTHETIC CONTRAST ENHANCED RADIOLOGICAL RECORDINGS Bayer Aktiengesellschaft (DE) 2025-12-17 EP claimed
EP-4475137-B1 GENERATION OF ARTIFICIAL CONTRAST ENHANCED RADIOLOGICAL RECORDINGS BAYER AG (DE) 2025-12-03 EP claimed
EP-4567715-A1 GENERATING SYNTHETIC REPRESENTATIONS Bayer Aktiengesellschaft (DE) 2025-06-11 EP claimed
EP-4498324-A1 DETECTING ARTIFACTS IN SYNTHETIC IMAGES Bayer AG (DE) 2025-01-29 EP claimed
EP-4485474-A2 GENERATION OF ARTIFICIAL CONTRAST ENHANCED RADIOLOGICAL RECORDINGS Bayer AG (DE) 2025-01-01 EP claimed
EP-4475137-A1 GENERATION OF ARTIFICIAL CONTRAST ENHANCED RADIOLOGICAL RECORDINGS Bayer AG (DE) 2024-12-11 EP claimed
WO-2024100233-A1 GENERATION OF ARTIFICIAL CONTRAST-ENHANCED RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-05-16 WO claimed
WO-2024052156-A1 GENERATION OF ARTIFICIAL CONTRAST-ENHANCED RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-14 WO claimed
WO-2024052549-A1 NEW CONTRAST AGENTS FOR USE IN DIAGNOSTIC IMAGING BAYER AKTIENGESELLSCHAFT (DE) 2024-03-14 WO claimed
EP-4335840-A1 NEW CONTRAST AGENTS FOR USE IN DIAGNOSTIC IMAGING Bayer Aktiengesellschaft (DE) 2024-03-13 EP claimed
WO-2024046832-A1 GENERATION OF SYNTHETIC RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-07 WO claimed
WO-2024046831-A1 GENERATION OF SYNTHETIC RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-07 WO claimed
WO-2024046833-A1 GENERATION OF SYNTHETIC RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-07 WO claimed
EP-4567716-B1 GENERATING SYNTHETIC REPRESENTATIONS BAYER AG (DE) 2026-05-13 EP disclosed
EP-4567715-B1 GENERATING SYNTHETIC REPRESENTATIONS BAYER AG (DE) 2026-05-13 EP disclosed
EP-4581641-B1 GENERATION OF SYNTHETIC RADIOLOGICAL RECORDINGS BAYER AG (DE) 2026-05-06 EP disclosed
EP-4581640-B1 GENERATION OF SYNTHETIC RADIOLOGICAL RECORDINGS BAYER AG (DE) 2026-04-22 EP disclosed
EP-4485474-B1 GENERATION OF ARTIFICIAL CONTRAST ENHANCED RADIOLOGICAL RECORDINGS BAYER AG (DE) 2026-04-08 EP disclosed
US-20260051027-A1 GENERATION OF SYNTHETIC CONTRAST-ENHANCED RADIOLOGICAL IMAGES BAYER AG (DE) 2026-02-19 US disclosed
EP-4664393-A1 GENERATION OF SYNTHETIC CONTRAST ENHANCED RADIOLOGICAL RECORDINGS Bayer Aktiengesellschaft (DE) 2025-12-17 EP disclosed
EP-4475137-B1 GENERATION OF ARTIFICIAL CONTRAST ENHANCED RADIOLOGICAL RECORDINGS BAYER AG (DE) 2025-12-03 EP disclosed
EP-4567716-A1 GENERATING SYNTHETIC REPRESENTATIONS Bayer Aktiengesellschaft (DE) 2025-06-11 EP disclosed
EP-4567715-A1 GENERATING SYNTHETIC REPRESENTATIONS Bayer Aktiengesellschaft (DE) 2025-06-11 EP disclosed
EP-4498324-A1 DETECTING ARTIFACTS IN SYNTHETIC IMAGES Bayer AG (DE) 2025-01-29 EP disclosed
EP-4485474-A2 GENERATION OF ARTIFICIAL CONTRAST ENHANCED RADIOLOGICAL RECORDINGS Bayer AG (DE) 2025-01-01 EP disclosed
EP-4475137-A1 GENERATION OF ARTIFICIAL CONTRAST ENHANCED RADIOLOGICAL RECORDINGS Bayer AG (DE) 2024-12-11 EP disclosed
EP-4375919-A1 GENERATION OF CONTRAST ENHANCED SYNTHETIC RADIOLOGICAL RECORDINGS Bayer AG (DE) 2024-05-29 EP disclosed
WO-2024100233-A1 GENERATION OF ARTIFICIAL CONTRAST-ENHANCED RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-05-16 WO disclosed
EP-4369353-A1 GENERATION OF ARTIFICIAL CONTRAST AGENT-ENHANCED RADIOLOGICAL RECORDINGS Bayer Aktiengesellschaft (DE) 2024-05-15 EP disclosed
WO-2024083466-A1 AUTOMATED ANALYSIS OF RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-04-25 WO disclosed
WO-2024052573-A1 COMBINATIONS OF CONTRAST AGENTS BAYER AKTIENGESELLSCHAFT (DE) 2024-03-14 WO disclosed
WO-2024052156-A1 GENERATION OF ARTIFICIAL CONTRAST-ENHANCED RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-14 WO disclosed
WO-2024052549-A1 NEW CONTRAST AGENTS FOR USE IN DIAGNOSTIC IMAGING BAYER AKTIENGESELLSCHAFT (DE) 2024-03-14 WO disclosed
EP-4335840-A1 NEW CONTRAST AGENTS FOR USE IN DIAGNOSTIC IMAGING Bayer Aktiengesellschaft (DE) 2024-03-13 EP disclosed
EP-4335461-A1 COMBINATIONS OF CONTRAST AGENTS Bayer AG (DE) 2024-03-13 EP disclosed
WO-2024046832-A1 GENERATION OF SYNTHETIC RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-07 WO disclosed
WO-2024046832-A1 GENERATION OF SYNTHETIC RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-07 WO disclosed
WO-2024046831-A1 GENERATION OF SYNTHETIC RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-07 WO disclosed
WO-2024046833-A1 GENERATION OF SYNTHETIC RADIOLOGICAL IMAGES BAYER AKTIENGESELLSCHAFT (DE) 2024-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260051027-A1 GENERATION OF SYNTHETIC CONTRAST-ENHANCED RADIOLOGICAL IMAGES WFS1, RXFP4, SLC11A2 MEN1 994/4885KMT2A 2963/4885FOLH1 2449/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.