SCHEMBL27172452

SCHEMBL27172452

CC(=O)C(=O)N1CC2CC(C1)C2NC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 9/20 0.41
CYP2C9 P11712 1/20 0.41
NR1H2 P55055 1/20 0.39
CTSK P43235 2/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
BTK Q06187 1/20 0.38
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
GAA P10253 1/20 0.35
RET P07949 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27172355 0.84 HSD11B1 (0.37) HSD11B1CYP2C9NR1H2CTSKCA1
SCHEMBL25694410 0.81 CTSK (0.42) HSD11B1CYP2C9NR1H2CTSKCA1
SCHEMBL20069820 0.81 CTSK (0.42) HSD11B1CYP2C9NR1H2CTSKCA1
SCHEMBL14657161 0.81 BTK (0.49) HSD11B1CYP2C9CTSKBTKNFKB1
SCHEMBL24091122 0.80 CTSK (0.41) HSD11B1CYP2C9NR1H2CTSKCA1
SCHEMBL30060502 0.78 EPHX2 (0.33) HSD11B1
SCHEMBL20413606 0.78 CTSK (0.40) HSD11B1CYP2C9NR1H2CTSKCA1
SCHEMBL20147716 0.78 CTSK (0.40) HSD11B1CYP2C9CTSKCA1CA2
SCHEMBL31644391 0.78 CTSK (0.40) HSD11B1CYP2C9NR1H2CTSKCA1
SCHEMBL20069821 0.78 CTSK (0.40) HSD11B1CYP2C9NR1H2CTSKCA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4339193-A1 COMPOUND HAVING ANTI-TUMOR ACTIVITY AND USE THEREOF Innovstone Therapeutics Limited (CN) 2024-03-20 EP disclosed
WO-2022237858-A1 COMPOUND HAVING ANTI-TUMOR ACTIVITY AND USE THEREOF 上海翊石医药科技有限公司 2022-11-17 WO disclosed