SCHEMBL27174693

SCHEMBL27174693

CN1CCN(c2ccc(Nc3ncc4ccccc4n3)cc2)CC1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP4K1 Q92918 1/20 0.73
EGFR P00533 6/20 0.66
ALK Q9UM73 2/20 0.65
CDK4 P11802 5/20 0.61
CCND3 P30281 4/20 0.61
CCND1 P24385 3/20 0.61
CCND2 P30279 3/20 0.61
AURKA O14965 2/20 0.60
ADRA2A P08913 2/20 0.60
ADRA2B P18089 2/20 0.60
ADRA2C P18825 2/20 0.60
KDM1A O60341 1/20 0.60
GLA P06280 1/20 0.60
SLC2A1 P11166 1/20 0.60
RECQL P46063 1/20 0.60
BLM P54132 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
CCNA2 P20248 2/20 0.59
CDK2 P24941 2/20 0.59
CCNK O75909 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29371810 0.86 KDM1A (0.62) MAP4K1EGFRALKCDK4CCND3
SCHEMBL29368254 0.86 MAP4K1 (0.60) MAP4K1EGFRALKAURKACCNA2
SCHEMBL29576526 0.85 WEE1 (0.56) MAP4K1EGFRALKCDK4CCND3
SCHEMBL29576898 0.85 HTR3A (0.68) MAP4K1EGFRALKCDK4CCND3
SCHEMBL29372589 0.84 ALK (0.67) EGFRALKCDK4CCND1CDK2
SCHEMBL29575732 0.84 SYK (0.56) MAP4K1EGFRALKCDK4CCND3
SCHEMBL29575978 0.84 MAP4K1 (0.55) MAP4K1EGFRALKCDK4CCND3
SCHEMBL29576356 0.84 JAK3 (0.56) MAP4K1EGFRALKCDK4CCND3
SCHEMBL29576068 0.84 MAP4K1 (0.72) MAP4K1EGFRALKCDK4CCND3
SCHEMBL29576631 0.83 MAP4K1 (0.54) MAP4K1EGFRALKCDK4CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260102406-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA INC (US) 2026-04-16 US disclosed
US-12403145-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC (US) 2025-09-02 US disclosed
US-20240197752-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA INC 2024-06-20 US disclosed
US-20240092761-A1 QUINAZOLINE COMPOUNDS AND METHODS OF USE IAMBIC THERAPEUTICS, INC. 2024-03-21 US disclosed
US-11865120-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC. (US) 2024-01-09 US disclosed
US-20220354864-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY NEUPHARMA, INC. 2022-11-10 US disclosed
US-11304957-B2 Substituted quinazolines for inhibiting kinase activity NEUPHARMA, INC. (US) 2022-04-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240092761-A1 QUINAZOLINE COMPOUNDS AND METHODS OF USE CCNI, CDK3, CDK1 MAP4K1 529/4885EGFR 831/4885ALK 2531/4885
US-20240197752-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY DCK, ABL1, MAP4K2 MAP4K1 16/4885EGFR 518/4885ALK 692/4885
US-11865120-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 MAP4K1 16/4885EGFR 518/4885ALK 692/4885
US-12403145-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 MAP4K1 16/4885EGFR 518/4885ALK 692/4885
US-11304957-B2 Substituted quinazolines for inhibiting kinase activity DCK, ABL1, MAP4K2 MAP4K1 16/4885EGFR 518/4885ALK 692/4885
US-20220354864-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY DCK, ABL1, MAP4K2 MAP4K1 16/4885EGFR 518/4885ALK 692/4885
US-20260102406-A1 SUBSTITUTED QUINAZOLINES FOR INHIBITING KINASE ACTIVITY BRAF, TTK, MAP4K2 MAP4K1 25/4885EGFR 290/4885ALK 441/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.