SCHEMBL27200081

SCHEMBL27200081

COCCCOc1cc(Br)cnc1F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.34
KMT2A Q03164 2/20 0.34
L3MBTL1 Q9Y468 5/20 0.33
ALDH1A1 P00352 2/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
MAPT P10636 3/20 0.32
HPGD P15428 3/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
LMNA P02545 2/20 0.32
SLC6A4 P31645 1/20 0.32
RECQL P46063 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
MET P08581 1/20 0.31
KDM1A O60341 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31365225 1.00 KDM4E (0.34) KDM4EKMT2AL3MBTL1ALDH1A1MEN1
SCHEMBL31365213 1.00 KDM4E (0.34) KDM4EKMT2AL3MBTL1ALDH1A1MEN1
SCHEMBL611267 0.83 PIK3CA (0.36) KDM4EKMT2AL3MBTL1ALDH1A1MEN1
SCHEMBL23884015 0.83 EGFR (0.33) KMT2AALDH1A1NPC1RAB9AMAPT
SCHEMBL19953240 0.80 KDM4E (0.39) KDM4EKMT2AL3MBTL1ALDH1A1MEN1
SCHEMBL18397199 0.79 GRM5 (0.44) KDM4EKMT2AL3MBTL1MEN1HPGD
SCHEMBL2118826 0.78 ALDH1A1 (0.40) KMT2AALDH1A1MEN1NPC1RAB9A
SCHEMBL29483025 0.78 ALDH1A1 (0.40) KMT2AALDH1A1MEN1NPC1RAB9A
SCHEMBL188937 0.75 PIK3CA (0.37) L3MBTL1SLC6A4KDM1A
SCHEMBL16930021 0.75 SLC6A4 (0.37) KDM4EKMT2AL3MBTL1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025008288-A1 9-OXO-9,10-DIHYDRO-6H-PYRANO[3,2-B:4,5-B']DIPYRIDINE-8-CARBOXYLIC ACID DERIVATIVES CENTENARA LABS AG (CH) 2025-01-09 WO disclosed
US-11964986-B1 9-oxo-9,10-dihydro-6H-pyrano[3,2-b:4,5-b′]dipyridine-8-carboxylic acid derivatives REJUVERON TELOMERE THERAPEUTICS AG (CH) 2024-04-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11964986-B1 9-oxo-9,10-dihydro-6H-pyrano[3,2-b:4,5-b′]dipyridine-8-carboxylic acid derivatives DPP9, DPYD, QDPR KDM4E 1901/4885KMT2A 3581/4885L3MBTL1 4763/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.