SCHEMBL27209658

SCHEMBL27209658

O=C(O)N1CCC(=Cc2cccc(Oc3cc(O)ccn3)c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FAAH O00519 13/20 0.47
CYP3A4 P08684 5/20 0.47
CYP2D6 P10635 4/20 0.47
GABRA1 P14867 1/20 0.47
ADRA2C P18825 1/20 0.47
CNR1 P21554 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
CNR2 P34972 1/20 0.47
HTR2B P41595 1/20 0.47
TMEM97 Q5BJF2 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
OGA O60502 2/20 0.39
LOX P28300 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
MGLL Q99685 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1011974 0.87 FAAH (0.54) FAAHCYP3A4CYP2D6GABRA1ADRA2C
SCHEMBL27094605 0.87 FAAH (0.51) FAAHCYP3A4CYP2D6GABRA1ADRA2C
SCHEMBL30657588 0.87 FAAH (0.51) FAAHCYP3A4CYP2D6GABRA1ADRA2C
SCHEMBL27209671 0.86 GPR119 (0.49) FAAHCYP3A4CYP2D6GABRA1ADRA2C
SCHEMBL27094609 0.83 CYP3A4 (0.49) FAAHCYP3A4CYP2D6GABRA1ADRA2C
SCHEMBL27209649 0.83 FAAH (0.45) FAAHCYP3A4CYP2D6GABRA1ADRA2C
SCHEMBL30903847 0.82 EPHX2 (0.49) FAAHCYP3A4CYP2D6GABRA1ADRA2C
SCHEMBL1012253 0.81 MGAM (0.48) OGA
SCHEMBL27094839 0.81 CYP3A4 (0.57) FAAHCYP3A4CYP2D6GABRA1ADRA2C
SCHEMBL1011754 0.80 FAAH (0.53) FAAHCYP3A4CYP2D6GABRA1ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240140930-A1 PIPERIDINE UREA DERIVATIVES FOR TREATMENT OF NEURODEGENERATIVE DISEASES NEUROPN THERAPEUTICS INC. (US) 2024-05-02 US disclosed
US-20240139172-A1 PIPERIDINE UREA DERIVATIVES FOR CANCER THERAPY NeuroPn Therapeutics, Inc. (US) 2024-05-02 US disclosed
WO-2024073648-A1 PIPERIDINE UREA DERIVATIVES FOR CANCER THERAPY NeuroPn Therapeutics, Inc. (US) 2024-04-04 WO disclosed
WO-2024073680-A1 PIPERIDINE UREA DERIVATIVES FOR TREATMENT OF NEURODEGENERATIVE DISEASES NEUROPN THERAPEUTICS INC. (US) 2024-04-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240139172-A1 PIPERIDINE UREA DERIVATIVES FOR CANCER THERAPY PDCD1, TP53, CHEK2 FAAH 3812/4885CYP3A4 3768/4885CYP2D6 4456/4885
US-20240140930-A1 PIPERIDINE UREA DERIVATIVES FOR TREATMENT OF NEURODEGENERATIVE DISEASES PRPH, EPHX1, BCHE FAAH 15/4885CYP3A4 2031/4885CYP2D6 3357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.