Amonafide

Amonafide

SCHEMBL27226

CN(C)CCN1C(=O)c2cccc3cc(N)cc(c23)C1=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 3/20 1.00
CYP2D6 P10635 1/20 1.00
POLB P06746 3/20 0.77
MEN1 O00255 2/20 0.77
KMT2A Q03164 2/20 0.77
NPSR1 Q6W5P4 2/20 0.77
CYP1A2 P05177 1/20 0.77
TNNI3 P19429 1/20 0.77
MAPK1 P28482 1/20 0.77
STAT6 P42226 1/20 0.77
TNNT2 P45379 1/20 0.77
TNNC1 P63316 1/20 0.77
HEXA P06865 5/20 0.74
HEXB P07686 5/20 0.74
PABPC1 P11940 1/20 0.67
AHR P35869 2/20 0.64
MAPT P10636 1/20 0.64
RECQL P46063 1/20 0.64
RAB9A P51151 1/20 0.64
LCK P06239 2/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Amonafide SCHEMBL29352008 1.00 FTO (1.00) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL6255345 1.00 FTO (1.00) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL1049714 0.99 FTO (0.97) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL1566668 0.99 FTO (0.97) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL1051955 0.99 FTO (0.97) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL20242315 0.94 FTO (0.88) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL1566374 0.93 FTO (0.86) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL9144516 0.93 FTO (0.86) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL1565520 0.93 FTO (0.86) FTOCYP2D6POLBMEN1KMT2A
Amonafide SCHEMBL5164837 0.92 FTO (0.84) FTOCYP2D6POLBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 8653 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137806-A1 INTERCALATING SUGAR MOLECULES XALUD THERAPEUTICS, INC. (US) 2026-05-21 US claimed
US-20260137707-A1 METHODS OF MODULATING ATXN2 EXPRESSION UNIV OF UTAH RESEARCH FOUNDATION (US) 2026-05-21 US claimed
US-20250275946-A1 COMBINATION THERAPY FOR THE TREATMENT OF CANCER UNM RAINFOREST INNOVATIONS (US) 2025-09-04 US claimed
EP-4608801-A1 ANTICANCER DRUG CONJUGATES Ariel Scientific Innovations Ltd. (IL) 2025-09-03 EP claimed
WO-2025129074-A2 INDEXING TECHNIQUES FOR TAGMENTED DNA LIBRARIES ILLUMINA, INC. (US) 2025-06-19 WO claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
EP-4536236-A2 METHODS OF MODULATING ATXN2 EXPRESSION University of Utah Research Foundation (US) 2025-04-16 EP claimed
EP-4525855-A1 INTERCALATING SUGAR MOLECULES Xalud Therapeutics, Inc. (US) 2025-03-26 EP claimed
CN-119285689-A Galactoside antitumor prodrug intermediate, and preparation and application thereof 江南大学 2025-01-10 CN claimed
WO-2024254465-A2 METHODS FOR PROMOTING EXPANSION OF HUMAN CD34+ CELLS IN VIVO AND FOR PROMOTING NEURAL REGENERATION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-12-12 WO claimed
WO-1995004757-A1 USE OF MONOCLONAL ANTIBODIES FOR DETERMINING SENSITIVITY TO ACETYLIZABLE DRUGS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1995-02-16 WO claimed
EP-0482043-B1 Monohydrochloride and monomethansulphonate of amonafide. KNOLL AG (DE) 1994-09-28 EP claimed
EP-0393575-B1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent SEARLE & CO (US) 1994-03-16 EP claimed
EP-0359347-B1 COVALENTLY-LINKED COMPLEXES AND METHODS FOR ENHANCED CYTOTOXICITY AND IMAGING NEORX CORPORATION (US) 1992-12-23 EP claimed
EP-0482043-A1 Monohydrochloride and monomethansulphonate of amonafide. KNOLL AG (DE) 1992-04-29 EP claimed
US-5057304-A Anticarcinogenic agents BASF AKTIENGESELLSCHAFT (DE) 1991-10-15 US claimed
EP-0443569-A2 Diamine derivatives and their use in oncology F. HOFFMANN-LA ROCHE AG (CH) 1991-08-28 EP claimed
WO-1991000857-A1 AMONAFIDE SALTS KNOLL AKTIENGESELLSCHAFT (DE) 1991-01-24 WO claimed
EP-0393575-A1 Neoplasia treatment compositions containing antineoplastic agent and side-effect reducing protective agent G.D. Searle & Co. (US) 1990-10-24 EP claimed
EP-0359347-A2 Covalently-linked complexes and methods for enhanced cytotoxicity and imaging NEORX CORPORATION (US) 1990-03-21 EP claimed