SCHEMBL2722809

SCHEMBL2722809

C/C=C/CN(Cc1ccccc1)C(C)=O

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.49
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
TDP1 Q9NUW8 1/20 0.45
CHRM2 P08172 1/20 0.45
CHRM4 P08173 1/20 0.45
CHRM5 P08912 1/20 0.45
CHRM1 P11229 1/20 0.45
CHRM3 P20309 1/20 0.45
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
TSPO P30536 1/20 0.43
TSHR P16473 2/20 0.42
FOLH1 Q04609 1/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2117209 0.82 LMNA (0.62) LMNANPC1RAB9ATDP1CHRM2
SCHEMBL24992390 0.81 NPSR1 (0.44) LMNANPC1RAB9ATDP1KMT2A
SCHEMBL24992374 0.81 NPSR1 (0.44) LMNANPC1RAB9ATDP1KMT2A
SCHEMBL7503719 0.81 LMNA (0.50) LMNANPC1RAB9ATDP1CHRM2
SCHEMBL11076827 0.77 HPGD (0.51) KMT2AMEN1ALDH1A1TSHR
SCHEMBL3836681 0.77 LMNA (0.72) LMNANPC1CHRM2CHRM4CHRM5
SCHEMBL1059560 0.77 LMNA (0.56) LMNANPC1RAB9ATDP1CHRM2
SCHEMBL5497633 0.75 ALDH1A1 (0.43) NPC1RAB9AKMT2AALDH1A1TSHR
SCHEMBL11378089 0.75 LMNA (0.55) LMNANPC1RAB9ATDP1CHRM2
SCHEMBL5073289 0.74 TSHR (0.46) NPC1RAB9AALDH1A1TSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2445878-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO Boehringer Ingelheim International GmbH (DE) 2012-05-02 EP disclosed
WO-2010149684-A1 NEW COMPOUNDS, PHARMACEUTICAL COMPOSITION AND METHODS RELATING THERETO BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-12-29 WO disclosed