SCHEMBL27235504

SCHEMBL27235504

COc1ccc(C)c(N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NNMT P40261 3/20 0.46
CYP1A2 P05177 1/20 0.46
KMT2A Q03164 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
NOS2 P35228 2/20 0.39
POLB P06746 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
DHFR P00374 1/20 0.38
PDE10A Q9Y233 2/20 0.37
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PIK3CA P42336 2/20 0.36
MTOR P42345 1/20 0.36
HTT P42858 1/20 0.35
TLR8 Q9NR97 1/20 0.34
CYP2A6 P11509 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29424844 0.81 NNMT (0.41) NNMTCYP1A2KMT2ASIRT2SIRT1
SCHEMBL126903 0.81 NNMT (0.41) NNMTCYP1A2KMT2ASIRT2SIRT1
Hydrochloric Acid SCHEMBL30078498 0.79 NNMT (0.40) NNMTCYP1A2KMT2ASIRT2SIRT1
Hydrochloric Acid SCHEMBL3338097 0.79 NNMT (0.40) NNMTCYP1A2KMT2ASIRT2SIRT1
SCHEMBL30884721 0.79 TLR8 (0.46) NNMTCYP1A2KMT2ASIRT2SIRT1
Hydrochloric Acid SCHEMBL3736737 0.79 NNMT (0.40) NNMTCYP1A2KMT2ASIRT2SIRT1
SCHEMBL172558 0.78 NNMT (0.52) NNMTCYP1A2KMT2ASIRT2SIRT1
SCHEMBL509468 0.77 NNMT (0.39) NNMTCYP1A2KMT2ASIRT2SIRT1
SCHEMBL2317842 0.77 SIRT2 (0.43) NNMTCYP1A2KMT2ASIRT2SIRT1
SCHEMBL30427669 0.77 NNMT (0.43) NNMTCYP1A2KMT2ASIRT2SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106660993-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2017-05-10 CN claimed
CN-106660993-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2017-05-10 CN disclosed