SCHEMBL27260720

SCHEMBL27260720

CS(=O)(=O)c1cccc(-c2ccnc3cc(-c4cnc(N)nc4)oc23)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.42
NR1H2 P55055 3/20 0.42
NR1H3 Q13133 3/20 0.42
ALOX5AP P20292 1/20 0.41
JAK2 O60674 1/20 0.41
ROCK1 Q13464 1/20 0.41
PIK3CA P42336 1/20 0.41
PIK3CB P42338 1/20 0.41
ATR Q13535 3/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
MAP3K7 O43318 1/20 0.39
TAB1 Q15750 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.38
CYP2C9 P11712 1/20 0.38
SYK P43405 1/20 0.37
RXRA P19793 1/20 0.37
PRKDC P78527 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27260619 0.89 NR1H2 (0.41) MTORNR1H2NR1H3ALOX5APJAK2
SCHEMBL27260990 0.83 NR1H2 (0.42) NR1H2NR1H3CYP2C9SYKRXRA
SCHEMBL27260814 0.83 NR1H2 (0.42) NR1H2NR1H3CYP2C9SYKRXRA
SCHEMBL27260617 0.82 KCNH2 (0.47) NR1H2NR1H3MAP3K7TAB1LOXL2
SCHEMBL722404 0.80 PDE4C (0.46) NR1H2NR1H3JAK2CA1CA2
SCHEMBL724751 0.80 MAP3K7 (0.47) NR1H2NR1H3MAP3K7TAB1LOXL2
SCHEMBL30765233 0.78 MAP3K7 (0.39) MTORNR1H2NR1H3JAK2PIK3CB
SCHEMBL30765322 0.78 FYN (0.41) NR1H2NR1H3ATRMAP3K7TAB1
SCHEMBL27260622 0.78 NR1H2 (0.38) MTORNR1H2NR1H3JAK2PIK3CB
SCHEMBL27260722 0.76 NR1H2 (0.43) NR1H2NR1H3JAK2SYKRXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024033280-A1 FUROPYRIDIN AND FUROPYRIMIDIN, INHIBITORS OF PI4K, FOR USE IN THE TREATMENT OF PARASITE INFECTION AND MALARIA MERCK PATENT GMBH (DE) 2024-02-15 WO disclosed