SCHEMBL30765322

SCHEMBL30765322

CN(C)CCOc1ccc(-c2cc3nccc(-c4cccc(S(C)(=O)=O)c4)c3o2)cn1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FYN P06241 2/20 0.41
ACVR1B P36896 1/20 0.38
TGFBR1 P36897 1/20 0.38
TDO2 P48775 1/20 0.36
ACVR1 Q04771 1/20 0.36
NR1H2 P55055 2/20 0.36
NR1H3 Q13133 2/20 0.36
MELK Q14680 2/20 0.36
CHEK2 O96017 1/20 0.35
RIPK2 O43353 1/20 0.35
NOD2 Q9HC29 1/20 0.35
ATM Q13315 3/20 0.35
ATR Q13535 1/20 0.35
PAICS P22234 1/20 0.34
OXTR P30559 1/20 0.34
MAP3K7 O43318 1/20 0.34
TAB1 Q15750 1/20 0.34
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27260619 0.80 NR1H2 (0.41) ACVR1NR1H2NR1H3RIPK2NOD2
SCHEMBL27260720 0.78 MTOR (0.42) NR1H2NR1H3RIPK2NOD2ATM
SCHEMBL27260814 0.76 NR1H2 (0.42) ACVR1NR1H2NR1H3KCNH2
SCHEMBL27260990 0.76 NR1H2 (0.42) ACVR1NR1H2NR1H3KCNH2
SCHEMBL30765233 0.74 MAP3K7 (0.39) ACVR1NR1H2NR1H3ATMATR
SCHEMBL722404 0.74 PDE4C (0.46) FYNNR1H2NR1H3
SCHEMBL27260617 0.74 KCNH2 (0.47) ACVR1NR1H2NR1H3MAP3K7TAB1
SCHEMBL724751 0.72 MAP3K7 (0.47) ACVR1NR1H2NR1H3MAP3K7TAB1
SCHEMBL30765376 0.72 MAP3K7 (0.39) ACVR1NR1H2NR1H3ATMATR
SCHEMBL27260978 0.72 MAP3K7 (0.39) ACVR1NR1H2NR1H3ATMATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024033280-A1 FUROPYRIDIN AND FUROPYRIMIDIN, INHIBITORS OF PI4K, FOR USE IN THE TREATMENT OF PARASITE INFECTION AND MALARIA MERCK PATENT GMBH (DE) 2024-02-15 WO disclosed