SCHEMBL2726257

SCHEMBL2726257

Cc1csc(-c2c(C)cc(-c3ncco3)cc2C(N)=O)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 1/20 0.36
SMPD1 P17405 1/20 0.34
GLRA3 O75311 1/20 0.34
GLRB P48167 1/20 0.34
TGFBR1 P36897 3/20 0.34
EEF2K O00418 1/20 0.34
NPC1 O15118 1/20 0.33
HCRTR1 O43613 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HSD17B10 Q99714 1/20 0.33
S100A4 P26447 1/20 0.33
FABP4 P15090 1/20 0.33
FABP5 Q01469 1/20 0.33
ADORA2A P29274 5/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2726893 0.88 ADORA2A (0.36) PIK3CBGLRA3GLRBTGFBR1EEF2K
SCHEMBL2726265 0.85 TGFBR1 (0.38) PIK3CBGLRA3GLRBTGFBR1NPC1
SCHEMBL2728038 0.82 KDM4B (0.39) PIK3CBGLRA3GLRBTGFBR1NPC1
SCHEMBL2726899 0.82 ADORA2A (0.36) PIK3CBGLRA3GLRBTGFBR1NPC1
SCHEMBL2725903 0.81 PIK3CB (0.36) PIK3CBGLRA3GLRBTGFBR1HCRTR1
SCHEMBL2729187 0.81 CHEK2 (0.37) PIK3CBTGFBR1EEF2KNPC1RAB9A
SCHEMBL2728332 0.78 KDM4E (0.39) PIK3CBTGFBR1NPC1RAB9A
SCHEMBL3648919 0.78 PIK3CB (0.36) PIK3CBGLRA3GLRBNPC1ALDH1A1
SCHEMBL2728011 0.78 PDE10A (0.53) TGFBR1NPC1ALDH1A1SMN1; SMN2NPSR1
SCHEMBL2724726 0.77 PARP1 (0.39) PIK3CBGLRA3GLRBEDNRABRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed